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Pack Size | Price | Availability | Quantity |
---|---|---|---|
25 mg | $3,170 | 10-14 weeks | |
50 mg | $4,180 | 10-14 weeks | |
100 mg | $5,800 | 10-14 weeks |
Description | GNE-616 is a highly potent, metabolically stable, orally bioavailable, and subtype-selective Nav1.7 inhibitor (Ki: 0.79 nM, Kd: 0.38 nM for hNav1.7) for the treatment of chronic pain. |
In vitro | Site-directed mutagenesis is critical for the isoform selectivity profile of GNE-616. |
In vivo | GNE-616 shows robust activity in a Nav1.7-dependent inherited erythromelalgia (IEM) PK/PD model. |
Molecular Weight | 537.53 |
Formula | C24H23F4N5O3S |
Cas No. | 2349371-81-7 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year |
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