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IV-255
IV-255
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IV-255
Catalog No. T78202
IV-255 is a selective small molecule inhibitor of the BRG1 bromodomain, heightening DNA damage when administered with Temozolomide and Bleomycin. It also curtails the invasiveness of GBM cells and augments both Temozolomide-induced cell death and Temozolomide's apoptosis-inducing activity [1].
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 2 mg | $88 | 5 days |
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Product Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | IV-255 is a selective small molecule inhibitor of the BRG1 bromodomain, heightening DNA damage when administered with Temozolomide and Bleomycin. It also curtails the invasiveness of GBM cells and augments both Temozolomide-induced cell death and Temozolomide's apoptosis-inducing activity [1]. |
| Molecular Weight | 359.37 |
| Formula | C19H19F2N3O2 |
| Cas No. |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year |
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