Shopping Cart
- Remove All
![TargetMol](https://www.targetmol.com/storage/error/oops.webp)
Your shopping cart is currently empty
Pack Size | Price | Availability | Quantity |
---|---|---|---|
25 mg | $766 | 1-2 weeks | |
50 mg | $995 | 1-2 weeks | |
100 mg | $1,510 | 1-2 weeks |
Description | LDN-192960 hydrochloride is an inhibitor of Dual-specificity Tyrosine-regulated Kinase 2 (DYRK2) and Haspin, with IC50 values of 48 nM and 10 nM, respectively. |
Targets&IC50 | Haspin:10 nM , DYRK2:48 nM |
In vitro | LDN-192960 hydrochloride (10 μM) inhibits ten other kinases by ≥90%, with five being potently inhibited (IC50<1 μM), including CLK1 (IC50=0.21 μM), DYRK1A (IC50=0.10 μM), DYRK2 (IC50=2 nM), DYRK3 (IC50=19 nM), and PIM1 (IC50=0.72 μM)[1]. |
Molecular Weight | 401.35 |
Formula | C18H22Cl2N2O2S |
Cas No. | 2309172-48-1 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
Copyright © 2015-2024 TargetMol Chemicals Inc. All Rights Reserved.