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LTB4 antagonist 2
Catalog No. T78677Cas No. 2929239-85-8
LTB4 antagonist 2, a carboxamide-acid compound, serves as an antagonist to leukotriene B4 (LTB4) with potential anti-inflammatory properties, exhibiting high affinity for the LTB4 receptor and an inhibitory concentration (IC50) of 439 nM [1].
LTB4 antagonist 2
Catalog No. T78677Cas No. 2929239-85-8
LTB4 antagonist 2, a carboxamide-acid compound, serves as an antagonist to leukotriene B4 (LTB4) with potential anti-inflammatory properties, exhibiting high affinity for the LTB4 receptor and an inhibitory concentration (IC50) of 439 nM [1].
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 25 mg | $1,970 | 8-10 weeks | |
| 50 mg | $2,580 | 8-10 weeks | |
| 100 mg | $3,400 | 8-10 weeks |
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LY255283
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Product Introduction
Bioactivity
Chemical Properties
| Description | LTB4 antagonist 2, a carboxamide-acid compound, serves as an antagonist to leukotriene B4 (LTB4) with potential anti-inflammatory properties, exhibiting high affinity for the LTB4 receptor and an inhibitory concentration (IC50) of 439 nM [1]. |
| Targets&IC50 | LTB4:439 nM |
| In vitro | LTB4 antagonist 2 (compound 24c), at concentrations of 0.1 μM and 10 μM, exhibits a specific binding inhibition of LTB4, achieving inhibition rates of 25% and 95%, respectively [1]. |
| Molecular Weight | 445.46 |
| Formula | C26H23NO6 |
| Cas No. | 2929239-85-8 |
Storage & Solubility Information
| Storage | Shipping with blue ice. |
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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