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PROTAC CDK9 degrader 4

Name: PROTAC CDK9 degrader 4
Brand: TargetMol
SKU: T39996
Price: 322 USD
Availability: InStock
Rating: 5 (10 reviews)

🥰Excellent

Catalog No. T39996Cas No. 2411021-01-5

PROTAC CDK9 degrader 4 is a highly potent CDK9 degrader that targets transcriptional regulation and has potential anticancer activity for the study of acute myelogenous leukemia (AML).

PROTAC CDK9 degrader 4

🥰Excellent

Catalog No. T39996Cas No. 2411021-01-5

PROTAC CDK9 degrader 4 is a highly potent CDK9 degrader that targets transcriptional regulation and has potential anticancer activity for the study of acute myelogenous leukemia (AML).

Pack Size	Price	Availability
1 mg	$322	In Stock
5 mg	$793	In Stock
10 mg	$1,280	In Stock
25 mg	$1,880	In Stock

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COA

All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

Product Introduction

Bioactivity

Description

PROTAC CDK9 degrader 4 is a highly potent CDK9 degrader that targets transcriptional regulation and has potential anticancer activity for the study of acute myelogenous leukemia (AML).

Chemical Properties

Molecular Weight	792.97
Formula	C₄₃H₅₆N₁₀O₅
Cas No.	2411021-01-5
Smiles	N(CC1=CC=C(NC(=O)N2CCN(CCCCCC3=C4C(C(=O)N(C4)C5C(=O)NC(=O)CC5)=CC=C3)CC2)C=C1)C=6N7C(=C(C(C)C)C=N7)N=C(N[C@@H](CC)CO)C6

Storage & Solubility Information

Storage

keep away from direct sunlight,keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

Solubility Information

DMSO: 80 mg/mL (100.89 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	1.2611 mL	6.3054 mL	12.6108 mL	63.0541 mL
5 mM	0.2522 mL	1.2611 mL	2.5222 mL	12.6108 mL
10 mM	0.1261 mL	0.6305 mL	1.2611 mL	6.3054 mL
20 mM	0.0631 mL	0.3153 mL	0.6305 mL	3.1527 mL
50 mM	0.0252 mL	0.1261 mL	0.2522 mL	1.2611 mL
100 mM	0.0126 mL	0.0631 mL	0.1261 mL	0.6305 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc