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AM12 inhibits lanthanide-evoked TRPC5 activity (IC50: 0.28 μM).
Pack Size | Price | Availability | Quantity |
---|---|---|---|
10 mg | $475 | 35 days | |
50 mg | $1,990 | 35 days |
Description | AM12 inhibits lanthanide-evoked TRPC5 activity (IC50: 0.28 μM). |
Targets&IC50 | TRPC5:0.28 μM |
In vitro | AM12 inhibits TRPC5 and TRPC4 channel activities evoked by the agonist (-)-Englerin A via a site accessible from the extracellular face of the membrane, acting directly on either the channel or a closely associated site. It also inhibits Ca2+ entry evoked by Gd3+, with an IC50 of 0.28 μM, demonstrating slightly higher potency than the natural product Galangin. |
Molecular Weight | 349.13 |
Formula | C15H9BrO5 |
Cas No. | 2387510-84-9 |
Relative Density. | 1.864 g/cm3 (Predicted) |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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