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DMT1 blocker 1

Catalog No. T11063   CAS 1354790-56-9

DMT1 blocker 1 is a blocker of divalent metal transporter 1 (DMT1) with IC50 of 0.64 μM, which is expected to block the absorption of iron by intestinal cells in vivo.

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DMT1 blocker 1 Chemical Structure
DMT1 blocker 1, CAS 1354790-56-9
Pack Size Availability Price/USD Quantity
1 mg In stock $ 135.00
5 mg In stock $ 289.00
10 mg In stock $ 478.00
25 mg In stock $ 789.00
50 mg In stock $ 1,080.00
100 mg In stock $ 1,480.00
500 mg In stock $ 2,970.00
1 mL * 10 mM (in DMSO) In stock $ 443.00
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Purity: 100%
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Biological Description
Chemical Properties
Storage & Solubility Information
Description DMT1 blocker 1 is a blocker of divalent metal transporter 1 (DMT1) with IC50 of 0.64 μM, which is expected to block the absorption of iron by intestinal cells in vivo.
Targets&IC50 DMT1 blocker 1:0.64 μM
Molecular Weight 294.31
Formula C16H14N4O2
CAS No. 1354790-56-9

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 45mg/mL (152.9mM), sonification is recommended.

TargetMolReferences and Literature

1. Cadieux JA, et al. Synthesis and biological evaluation of substituted pyrazoles as blockers of divalent metal transporter 1 (DMT1). Bioorg Med Chem Lett. 2012 Jan 1;22(1):90-5.

Related compound libraries

This product is contained In the following compound libraries:
Inhibitor Library Bioactive Compound Library Bioactive Compounds Library Max

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Keywords

DMT1 blocker 1 1354790-56-9 Others DMT-1 blocker 1 inhibitor inhibit

 

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