Powder: -20°C for 3 years | In solvent: -80°C for 1 year
MSOP is a selective antagonist of group III metabotropic glutamate receptor (KD of 51 μM for the L-AP4-sensitive presynaptic mGluR).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | 6-8 weeks | $ 987.00 | |
50 mg | 6-8 weeks | $ 1,340.00 | |
100 mg | 6-8 weeks | $ 1,990.00 |
Description | MSOP is a selective antagonist of group III metabotropic glutamate receptor (KD of 51 μM for the L-AP4-sensitive presynaptic mGluR). |
Targets&IC50 | L-AP4-sensitive presynaptic mGluR:(kd)51 μM |
In vivo | Intrathecal TBOA (10 μg) reduces the number of formalin-induced flinches and shakes by 47% of the value in the saline-treated group in the second phase (P<0.001) and blocked the CFA-induced decrease in ipsilateral paw withdrawal latency by 60% of the value in the saline-treated group (P=0.01).?The number of formalin-induced flinches in the second phase in the group treated with MSOP and TBOA is increased by 56% (P=0.04) of the value in the TBOA-treated group.?CFA-induced paw withdrawal latency in the group treated with MSOP and TBOA is decreased by 86% (P=0.03) of the value in the TBOA-treated group. |
Molecular Weight | 199.1 |
Formula | C4H10NO6P |
CAS No. | 66515-29-5 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. More
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MSOP 66515-29-5 Neuroscience GluR inhibitor inhibit