Powder: -20°C for 3 years | In solvent: -80°C for 1 year
PDE5-IN-2 is a potent, highly selective, and orally active inhibitor of PDE5(IC50 of 0.31 nM)
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | 8-10 weeks | $ 1,970.00 | |
50 mg | 8-10 weeks | $ 2,580.00 | |
100 mg | 8-10 weeks | $ 3,400.00 |
Description | PDE5-IN-2 is a potent, highly selective, and orally active inhibitor of PDE5(IC50 of 0.31 nM) |
Targets&IC50 | PDE5A1:0.31 nM, PDE2A:106 nM, PDE4D2:43 nM, PDE6C:1.2 nM, PDE10A:46 nM |
In vitro | PDE5-IN-2 has at least 1000-fold selectivity over PDE1B, PDE3A, PDE7A1, PDE8A1, and PDE9A2 (IC50s, >32 000 nM)[1]. |
In vivo | PDE5-IN-2 shows anti-pulmonary arterial hypertension activity[1]. |
Molecular Weight | 491.52 |
Formula | C25H21N3O6S |
CAS No. | 2244517-61-9 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. More
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PDE5-IN-2 2244517-61-9 Metabolism PDE PDE5 IN 2 PDE5IN2 PDE-5-IN-2 inhibitor inhibit