Powder: -20°C for 3 years | In solvent: -80°C for 1 year
PIM1-IN-1 is a potent and highly selective inhibitor of PIM1/3(IC50s of 7, 5530 and 70 nM for PIM1, PIM2, and PIM3, respectively),with Antiproliferative and anti-cancer activity.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | 8-10 weeks | $ 1,140.00 | |
50 mg | 8-10 weeks | $ 1,490.00 | |
100 mg | 8-10 weeks | $ 2,360.00 |
Description | PIM1-IN-1 is a potent and highly selective inhibitor of PIM1/3(IC50s of 7, 5530 and 70 nM for PIM1, PIM2, and PIM3, respectively),with Antiproliferative and anti-cancer activity. |
Targets&IC50 | Pim1:7 nM, Pim3:70 nM, Pim2:5530 nM |
In vitro | PIM1-IN-1 induces apoptosis in SKMEL19 cells[1]. |
In vivo | PIM1-IN-1 shows cceptable clearance of 1.26 L/h/kg in BALB-C mice[1]. |
Molecular Weight | 474.56 |
Formula | C25H30N8O2 |
CAS No. | 1417630-95-5 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. More
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PIM1-IN-1 1417630-95-5 Chromatin/Epigenetic JAK/STAT signaling Pim PIM1 IN 1 PIM1IN1 PIM-1-IN-1 inhibitor inhibit