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Apalutamide-13C-d3
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Catalog No. TMIH-0092
Alias RN509-13C,d3, RN-509-13C,d3
Apalutamide-13C-d3 (RN-509-13C,d3) is a 13C and 2H-labeled version of Apalutamide. Apalutamide is an efficient androgen receptor (AR) antagonist used in the study of prostate diseases.
Apalutamide-13C-d3
😃Good
Catalog No. TMIH-0092Alias RN509-13C,d3, RN-509-13C,d3
Apalutamide-13C-d3 (RN-509-13C,d3) is a 13C and 2H-labeled version of Apalutamide. Apalutamide is an efficient androgen receptor (AR) antagonist used in the study of prostate diseases.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $728 | 7-10 days | |
| 5 mg | $2,600 | 7-10 days | |
| 10 mg | Inquiry | 7-10 days |
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Product Introduction
Bioactivity
Chemical Properties
| Description | Apalutamide-13C-d3 (RN-509-13C,d3) is a 13C and 2H-labeled version of Apalutamide. Apalutamide is an efficient androgen receptor (AR) antagonist used in the study of prostate diseases. |
| Targets&IC50 | AR:16 nM |
| Alias | RN509-13C,d3, RN-509-13C,d3 |
| Molecular Weight | 481.45 |
| Formula | 13C C20H12F4N5O2SD3 |
| Smiles | FC(F)(F)C1=C(C#N)N=CC(N2C(C3(CCC3)N(C4=CC(F)=C(C(N[13C]([2H])([2H])[2H])=O)C=C4)C2=S)=O)=C1 |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 40 mg/mL (83.08 mM), Sonication is recommended. | ||||||||||||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||||||||||||
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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