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Apalutamide-13C-d3

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Catalog No. TMIH-0092
Alias RN509-13C,d3, RN-509-13C,d3

Apalutamide-13C-d3 (RN-509-13C,d3) is a 13C and 2H-labeled version of Apalutamide. Apalutamide is an efficient androgen receptor (AR) antagonist used in the study of prostate diseases.

Apalutamide-13C-d3

Apalutamide-13C-d3

😃Good
Catalog No. TMIH-0092Alias RN509-13C,d3, RN-509-13C,d3
Apalutamide-13C-d3 (RN-509-13C,d3) is a 13C and 2H-labeled version of Apalutamide. Apalutamide is an efficient androgen receptor (AR) antagonist used in the study of prostate diseases.
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1 mg$728 7-10 days
5 mg$2,600 7-10 days
10 mgInquiry7-10 days
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Product Introduction

Bioactivity
Description
Apalutamide-13C-d3 (RN-509-13C,d3) is a 13C and 2H-labeled version of Apalutamide. Apalutamide is an efficient androgen receptor (AR) antagonist used in the study of prostate diseases.
Targets&IC50
AR:16 nM
AliasRN509-13C,d3, RN-509-13C,d3
Chemical Properties
Molecular Weight481.45
Formula13C C20H12F4N5O2SD3
SmilesFC(F)(F)C1=C(C#N)N=CC(N2C(C3(CCC3)N(C4=CC(F)=C(C(N[13C]([2H])([2H])[2H])=O)C=C4)C2=S)=O)=C1
Storage & Solubility Information
StorageShipping with blue ice.
Solubility Information
DMSO: 40 mg/mL (83.08 mM), Sonication is recommended.
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.0771 mL10.3853 mL20.7706 mL103.8529 mL
5 mM0.4154 mL2.0771 mL4.1541 mL20.7706 mL
10 mM0.2077 mL1.0385 mL2.0771 mL10.3853 mL
20 mM0.1039 mL0.5193 mL1.0385 mL5.1926 mL
50 mM0.0415 mL0.2077 mL0.4154 mL2.0771 mL

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Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
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