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EPZ020411 is a specific and effective inhibitor of PRMT6 (IC50=10 nM).
Pack Size | Price | Availability | Quantity |
---|---|---|---|
2 mg | 130 € | 5 days | |
5 mg | 223 € | 7-10 days | |
10 mg | 372 € | 7-10 days |
Description | EPZ020411 is a specific and effective inhibitor of PRMT6 (IC50=10 nM). |
Targets&IC50 | PRMT6:10 nM |
In vitro | In PRMT6-overexpressing cells, EPZ020411 does-dependently inhibits H3R2 methylation. |
In vivo | in vivo: EPZ020411 shows good bioavailability following subcutaneous (SC) dosing in rats making it a suitable tool for in vivo studies. |
Molecular Weight | 442.6 |
Formula | C25H38N4O3 |
Cas No. | 1700663-41-7 |
Smiles | CNCCN(C)Cc1c[nH]nc1-c1ccc(O[C@H]2C[C@@H](C2)OCCC2CCOCC2)cc1 |
Relative Density. | 1.16 g/cm3 (Predicted) |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||
Solubility Information | DMSO: 10 mM | ||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||
DMSO
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