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hGPR91 antagonist 3

Name: hGPR91 antagonist 3
Brand: TargetMol
SKU: T62858
Price: 149 USD
Availability: InStock
Rating: 5 (10 reviews)

🥰Excellent

Catalog No. T62858Cas No. 1314796-31-0

hGPR91 antagonist 3 is an orally active, potent, and selective hGPR91 antagonist. hGPR91 antagonist 3 is used to study hypertension, autoimmune diseases, and retinal angiogenesis. hGPR91 antagonist 3 has been shown to be effective in the treatment of hypertension, autoimmune disease, and retinal angiogenesis.

hGPR91 antagonist 3

🥰Excellent

Purity: 98.82%

Catalog No. T62858Cas No. 1314796-31-0

Pack Size	Price	Availability	Quantity
1 mg	$149	In Stock

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Purity:98.82%

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COA HNMR HPLC LCMS

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Product Introduction

Bioactivity

Description	hGPR91 antagonist 3 is an orally active, potent, and selective hGPR91 antagonist. hGPR91 antagonist 3 is used to study hypertension, autoimmune diseases, and retinal angiogenesis. hGPR91 antagonist 3 has been shown to be effective in the treatment of hypertension, autoimmune disease, and retinal angiogenesis.
Targets&IC50	GPR91:135 nM (Rat), GPR91 (human):35 nM

Chemical Properties

Molecular Weight	458.41
Formula	C₂₃H₁₈F₄N₄O₂
Cas No.	1314796-31-0
Smiles	O=C(NCC=1ON=C(C1)C=2C=CC(F)=C(C2)C(F)(F)F)CCCC=3N=C4N=CC=CC4=CC3

Storage & Solubility Information

Storage

store under nitrogen | Shipping with blue ice.

Solubility Information

DMSO: 80 mg/mL (174.52 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.1815 mL	10.9073 mL	21.8145 mL	109.0727 mL
5 mM	0.4363 mL	2.1815 mL	4.3629 mL	21.8145 mL
10 mM	0.2181 mL	1.0907 mL	2.1815 mL	10.9073 mL
20 mM	0.1091 mL	0.5454 mL	1.0907 mL	5.4536 mL
50 mM	0.0436 mL	0.2181 mL	0.4363 mL	2.1815 mL
100 mM	0.0218 mL	0.1091 mL	0.2181 mL	1.0907 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc