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NLRP3 agonist 1
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Catalog No. T81668Cas No. 2454019-69-1
NLRP3 agonist 1 is an orally active and highly potent NLRP3 agonist that activates the enzyme Caspase-1, which may promote the maturation of pro-inflammatory cytokines.
NLRP3 agonist 1
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Purity: 99.01%
Catalog No. T81668Cas No. 2454019-69-1
NLRP3 agonist 1 is an orally active and highly potent NLRP3 agonist that activates the enzyme Caspase-1, which may promote the maturation of pro-inflammatory cytokines.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 5 mg | Inquiry | In Stock | |
| 50 mg | Inquiry | 8-10 weeks |
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Purity:99.01%
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Product Introduction
Bioactivity
Chemical Properties
| Description | NLRP3 agonist 1 is an orally active and highly potent NLRP3 agonist that activates the enzyme Caspase-1, which may promote the maturation of pro-inflammatory cytokines. |
| Molecular Weight | 280.33 |
| Formula | C15H16N6 |
| Cas No. | 2454019-69-1 |
| Smiles | N=1NC=CC1C=2C=CC3=C(N=C(N=C3NC4(C)CC4)N)C2 |
Storage & Solubility Information
| Storage | store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 80 mg/mL (285.38 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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