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PROTAC Her3 Degrader-8
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Catalog No. T77976Cas No. 2103331-95-7
PROTAC Her3 Degrader-8 (Compound PP2) is a proteolysis targeting chimera (PROTAC) that degrades the Her3 protein in vitro and in cellular assays, with potential applications in investigating diseases modulated by HER family proteins [1].
PROTAC Her3 Degrader-8
😃Good
Catalog No. T77976Cas No. 2103331-95-7
PROTAC Her3 Degrader-8 (Compound PP2) is a proteolysis targeting chimera (PROTAC) that degrades the Her3 protein in vitro and in cellular assays, with potential applications in investigating diseases modulated by HER family proteins [1].
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Product Introduction
Bioactivity
Chemical Properties
| Description | PROTAC Her3 Degrader-8 (Compound PP2) is a proteolysis targeting chimera (PROTAC) that degrades the Her3 protein in vitro and in cellular assays, with potential applications in investigating diseases modulated by HER family proteins [1]. |
| Molecular Weight | 926.1 |
| Formula | C49H55N11O6S |
| Cas No. | 2103331-95-7 |
Storage & Solubility Information
| Storage | Shipping with blue ice. |
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DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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