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Bremelanotide Acetate

Catalog No. T7608 CAS 1607799-13-2

Synonyms: bremelanotide, PT-141 Acetate

Bremelanotide Acetate (PT-141 Acetate) is an agonist of melanocortin receptor (MCR) .

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

Bremelanotide Acetate Chemical Structure

Bremelanotide Acetate, CAS 1607799-13-2

Pack Size	Availability	Price/USD
10 mg	In stock	$ 46.00
25 mg	In stock	$ 83.00
50 mg	In stock	$ 139.00
100 mg	In stock	$ 207.00
1 mL * 10 mM (in DMSO)	In stock	$ 65.00

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Purity: 98%

Biological Description

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Description	Bremelanotide Acetate (PT-141 Acetate) is an agonist of melanocortin receptor (MCR) .
In vivo	Treatment with Bremelanotide?(100 or 200 μg/kg) significantly increased proceptive solicitations in females primed with E+Por E alone (E+O) in bilevel chambers[1]
Animal Research	Bremelanotide(PT-141), a cyclic heptapeptide melanocortin analogue (Palatin Technologies, Cranbury, NJ), was dissolved in saline to obtain doses of 50, 100, and 200 μg/kg/ml, and injected s.c. 5 min before each behavioral test. An equal volume of saline was administered to control animals[1].

Synonyms	bremelanotide, PT-141 Acetate
Molecular Weight	1085.22
Formula	C52H72N14O12
CAS No.	1607799-13-2

Storage

keep away from moisture

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 36 mg/mL (33.17 mM)

References and Literature

1. Pfaus JG, Shadiack A, Van Soest T,et al.Selective facilitation of sexual solicitation in the female rat by a melanocortin receptor agonist[J].Proc Natl Acad Sci U S A. 2004 Jul 6;101(27) 2. Clayton AH, Althof SE, Kingsberg S,et al.Bremelanotide for female sexual dysfunctions in premenopausal women: a randomized, placebo-controlled dose-finding trial[J].Womens Health (Lond). 2016 Jun;12(3):325-37.

Related compound libraries

This product is contained In the following compound libraries：

Peptide Compound Library Anti-Cancer Clinical Compound Library Drug Repurposing Compound Library Anti-Cancer Drug Library Anti-Cancer Approved Drug Library Neuronal Signaling Compound Library Clinical Compound Library Bioactive Compounds Library Max FDA-Approved Drug Library Anti-Cancer Compound Library

Related Products

Related compounds with same targets

TCMCB07 TFA JNJ-10229570 Setmelanotide Acetate(920014-72-8 free base) a-MSH, amide Acetate(581-05-5 free base) HS 014 acetate(207678-81-7 free base) AP1189 acetate α-MSH Undecylenoyl phenylalanine

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

Bremelanotide Acetate 1607799-13-2 GPCR/G Protein Neuroscience Melanocortin Receptor PT 141 Acetate bremelanotide inhibit PT141 PT141 Acetate PT-141 Acetate MC Receptor PT 141 Inhibitor PT-141 inhibitor

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