Powder: -20°C for 3 years | In solvent: -80°C for 1 year
CRTh2 antagonist 2 is a selective and potent CRTH2 antagonist, IC50≤10 nM. CRTh2 antagonist 2 can be used to study the direction of androgenic alopecia.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 183.00 | |
5 mg | In stock | $ 361.00 | |
10 mg | In stock | $ 587.00 | |
25 mg | In stock | $ 938.00 | |
50 mg | In stock | $ 1,280.00 | |
100 mg | In stock | $ 1,720.00 | |
500 mg | In stock | $ 3,450.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 483.00 |
Description | CRTh2 antagonist 2 is a selective and potent CRTH2 antagonist, IC50≤10 nM. CRTh2 antagonist 2 can be used to study the direction of androgenic alopecia. |
Targets&IC50 | CRTH2:≤10 nM |
In vitro | CRTH2, also known as GPR44(chemoattractant receptor-homologous molecule expressed on Th2 cells) protein, is a G-protein coupled receptor (GPCR) which is amongst other ligands most strongly activated by prostaglandin D2 (PGD2). PGD2 is a product of prostaglandin D2 synthase (PTGDS)[1]. |
Molecular Weight | 474.94 |
Formula | C26H23ClN4O3 |
CAS No. | 780763-95-3 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 45 mg/mL (94.75 mM)
You can also refer to dose conversion for different animals. More
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CRTh2 antagonist 2 780763-95-3 Endocrinology/Hormones GPCR/G Protein GPR CRTh-2 antagonist 2 inhibitor inhibit