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Antitumor agent-87

Antitumor agent-87 is a potent compound exhibiting high antitumoral activity, with a Ki value of 0.23 µM for CYP1A1. It demonstrates antiproliferative effects and induces cell cycle arrest at the G2/M phase, underscoring its effectiveness as an antitumor agent.

Catalog No. T72551Cas No. 1422527-88-5

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Purity:99.75%

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COA HNMR HPLC LCMS

Antitumor agent-87

Catalog No. T72551Cas No. 1422527-88-5

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Pack Size	Price	Availability
1 mg	$293	In Stock
5 mg	$722	In Stock
10 mg	$987	In Stock
25 mg	$1,520	In Stock
50 mg	$1,980	In Stock

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Product Introduction

Bioactivity

Description	Antitumor agent-87 is a potent compound exhibiting high antitumoral activity, with a Ki value of 0.23 µM for CYP1A1. It demonstrates antiproliferative effects and induces cell cycle arrest at the G2/M phase, underscoring its effectiveness as an antitumor agent.
Targets&IC50	CYP1A1:0.23 μM (Ki), M21:>12500 nM, MCF7:600 nM, MLKL (HT-29 cells):>12500 nM
In vitro	In MCF7, HT-29, and M21 cells, Antitumor agent-87 (0-12500 nM; 48 hours) exhibited antiproliferative activity with IC50 values of 600 nM, >12500 nM, and >12500 nM, respectively[1].
In vivo	Antitumor agent-87 ( 0.1μg/egg ) showed 29 % anti-tumor activity in transplanted HT-1080 chick embryos [1].

Chemical Properties

Molecular Weight	448.53
Formula	C₂₂H₂₈N₂O₆S
Cas No.	1422527-88-5

Storage & Solubility Information

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Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

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