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Melanostatin, frog TFA
🥰Excellent
Catalog No. TP2603L
Alias Melanostatin, frog TFA(134709-16-3 Free base)
Melanostatin, frog TFA is a highly efficient α-melanocyte-stimulating hormone (α-MSH) release inhibitor, a 36-amino acid peptide isolated from the frog brain, which modulates the electrophysiological activity of frog melanocytes by regulating K+, Na+, and Ca2+ currents.
Melanostatin, frog TFA
Melanostatin, frog TFA
🥰Excellent
Catalog No. TP2603LAlias Melanostatin, frog TFA(134709-16-3 Free base)
Melanostatin, frog TFA is a highly efficient α-melanocyte-stimulating hormone (α-MSH) release inhibitor, a 36-amino acid peptide isolated from the frog brain, which modulates the electrophysiological activity of frog melanocytes by regulating K+, Na+, and Ca2+ currents.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $195 | In Stock | |
| 5 mg | $582 | In Stock | |
| 10 mg | $829 | In Stock | |
| 25 mg | $1,260 | In Stock | |
| 50 mg | $1,680 | In Stock | |
| 100 mg | $2,280 | In Stock |
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Product Introduction
Bioactivity
Chemical Properties
| Description | Melanostatin, frog TFA is a highly efficient α-melanocyte-stimulating hormone (α-MSH) release inhibitor, a 36-amino acid peptide isolated from the frog brain, which modulates the electrophysiological activity of frog melanocytes by regulating K+, Na+, and Ca2+ currents. |
| Targets&IC50 | α-MSH:60 nM |
| In vitro | Melanostatin, frog TFA is a potent inhibitor of α-melanocyte-stimulating hormone (α-MSH) release with an IC50 value of 60 nM.At a concentration of 1 μM, Melanostatin, frog TFA enhances potassium currents, while decreasing sodium and calcium currents, thereby inducing hyperpolarization of the cell membrane. [1] |
| Alias | Melanostatin, frog TFA(134709-16-3 Free base) |
Storage & Solubility Information
| Storage | keep away from direct sunlight,keep away from moisture,store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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