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HS024

Catalog No. TP1898Cas No. 212370-59-7
Alias HS 024

HS024 is a highly potent melanocortin MC4 receptor antagonist (Ki values are 0.29, 18.6, 5.45 and 3.29 nM for cloned human MC4, MC1, MC3 and MC5 receptors respectively). Increases food intake, and blocks α-MSH- and MTII-induced hypotension and bradycardia in rats, following central administration in vivo.

HS024

HS024

Purity: 100%
Catalog No. TP1898Alias HS 024Cas No. 212370-59-7
HS024 is a highly potent melanocortin MC4 receptor antagonist (Ki values are 0.29, 18.6, 5.45 and 3.29 nM for cloned human MC4, MC1, MC3 and MC5 receptors respectively). Increases food intake, and blocks α-MSH- and MTII-induced hypotension and bradycardia in rats, following central administration in vivo.
Pack SizePriceAvailabilityQuantity
1 mg$346In Stock
5 mg$835In Stock
10 mg$1,150In Stock
25 mg$1,690In Stock
50 mg$2,290In Stock
100 mg$3,120In Stock
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Purity:100%
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Product Introduction

Bioactivity
Description
HS024 is a highly potent melanocortin MC4 receptor antagonist (Ki values are 0.29, 18.6, 5.45 and 3.29 nM for cloned human MC4, MC1, MC3 and MC5 receptors respectively). Increases food intake, and blocks α-MSH- and MTII-induced hypotension and bradycardia in rats, following central administration in vivo.
AliasHS 024
Chemical Properties
Molecular Weight1266.5
FormulaC58H79N19O10S2
Cas No.212370-59-7
Storage & Solubility Information
Storagekeep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
H2O: 0.50 mg/mL

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