Shopping Cart
- Remove All
Your shopping cart is currently empty
Bremelanotide Acetate
🥰Excellent
Catalog No. T7608Cas No. 1607799-13-2
Alias PT-141 Acetate
Bremelanotide Acetate (PT-141 Acetate) is an agonist of melanocortin receptor (MCR) .
Bremelanotide Acetate
🥰Excellent
Purity: 100.00%
Catalog No. T7608Alias PT-141 AcetateCas No. 1607799-13-2
Bremelanotide Acetate (PT-141 Acetate) is an agonist of melanocortin receptor (MCR) .
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 10 mg | $46 | In Stock | |
| 25 mg | $83 | In Stock | |
| 50 mg | $139 | In Stock | |
| 100 mg | $207 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $65 | In Stock |
Bulk & Custom
Add to Cart
Questions
View MoreInhibitors Related to "Bremelanotide Acetate"
Undecylenoyl phenylalanine
Undecylenoylphenylalanine, Sepiwhite msh QD
T20501175357-18-3
Undecylenoyl phenylalanine (Sepiwhite msh QD) is a novel depigmenting agent, which possibly acts as an alpha-melanocyte-stimulating hormone antagonist, thus inhibiting melaninogenesis.
- $29
Size
QTY
ACTH (1-17) acetate
TP1011L
ACTH (1-17) acetate is a potent agonist at the human melanocortin 1 (MC1) receptor with high affinity(Ki = 0.21 nM).
- $122
Size
QTY
[D-Trp8]-γ-MSH acetate(321351-81-9 free base)
TP1893L1
[D-Trp8]-γ-MSH acetate(321351-81-9 free base) is a selective melanocortin 3 (MC3) receptor agonist (IC50 values are 6.7, 340 and 600 nM for human MC3, MC5 and MC4 receptors respectively) and displays anti-inflammatory efficacy.
- $143
Size
QTY
Fenoprofen
Nalgesic, Nalfon
T0184L29679-58-1
Fenoprofen (LILLY-5385) is a non-steroidal anti-inflammatory compound and a modifier enhancer of the melanocortin receptor, which increases ERK1/2 activation, inhibits biofilm formation, and alters biofilm structure, and is used in the treatment of acute pain and chronic arthritis.
- $30
Size
QTY
HS 014 acetate(207678-81-7 free base)
TP2015L
HS 014 acetate is a potent and selective melanocortin MC4 receptor antagonist (Ki values are 3.16, 108, 54.4 and 694 nM for cloned human MC4, MC1, MC3 and MC5 receptors respectively). Increases food intake in rats and nociception in mice following central
- $185
Size
QTY
ACTH 11-24 acetate(4237-93-8 free base)
Adrenocorticotropic Hormone (11-24) acetate
TP1248L79190-56-0
ACTH 11-24 acetate(4237-93-8 free base) (Adrenocorticotropic Hormone (11-24) acetate) is a fragment of adrenocorticotrophin, induces cortisol release. ACTH (11-24) has been identified as a competitive antagonist of ACTH (1-39) and ACTH (1-10) in isolated adrenal cells.
- $44
Size
QTY
Neuropeptide EI, rat acetate
Neuropeptide EI, rat acetate(125934-45-4 free base)
TP1578L
Neuropeptide EI, rat acetate Displays functional MCH-antagonist and MSH-agonist activity in different behavioral paradigms.
- $65
Size
QTY
Beta-MSH (1-22) (human) acetate
Beta-MSH (1-22) (human) acetate (17908-57-5 Free base)
TP1004L
Beta-MSH (1-22) (human) acetate (Beta-MSH (1-22) (human) acetate (17908-57-5 Free base)) , is an endogenous melanocortin-4 receptor (MC4-R) agonist.
- $167
Size
QTY
HS024
HS 024
TP1898212370-59-7
HS024 is a highly potent melanocortin MC4 receptor antagonist (Ki values are 0.29, 18.6, 5.45 and 3.29 nM for cloned human MC4, MC1, MC3 and MC5 receptors respectively). Increases food intake, and blocks α-MSH- and MTII-induced hypotension and bradycardia in rats, following central administration in vivo.
- $346
Size
QTY
MCL0020
MCL 0020
TP1889475498-26-1
MCL0020 is a potent and selective melanocortin MC4 receptor antagonist (IC50 values are 11.63, 1115, and >10,000 nM at MC4, MC3, and MC1 receptors, respectively). It significantly reverses stress-induced anorexia without affecting food intake in free-feeding rats and exhibits anxiolytic-like activity in vivo.
- $118
Size
QTY
Nonapeptide-1 acetate salt (158563-45-2 free base)
Nonapeptide-1 acetate salt, Melanostatine-5 acetate salt
TP1101
Nonapeptide-1 acetate salt (158563-45-2 free base) (Melanostatine-5 acetate salt) , a peptide hormone, is a potent α-Melanocyte-stimulating hormone (α-MSH) antagonist, with an IC50 of 11 nM. Nonapeptide-1 acetate salt (158563-45-2 free base) , a peptide hormone, is a potent α-Melanocyte-stimulating hormone (α-MSH) antagonist, with an IC50 of 11 nM.
- $63
Size
QTY
α-MSH, amide Acetate
TP2212L
a-MSH, amide Acetate as an endogenous neuropeptide. It is an endogenous melanocortin receptor 4 (MC4R) agonist with anti-inflammatory and antipyretic activities. α-MSH is a post-translational derivative of pro-opiomelanocortin (POMC)
- $45
Size
QTY
Select Batch
Purity:100.00%
Contact us for more batch information
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Bremelanotide Acetate (PT-141 Acetate) is an agonist of melanocortin receptor (MCR) . |
| In vivo | Treatment with Bremelanotide?(100 or 200 μg/kg) significantly increased proceptive solicitations in females primed with E+Por E alone (E+O) in bilevel chambers[1] |
| Animal Research | Bremelanotide(PT-141), a cyclic heptapeptide melanocortin analogue (Palatin Technologies, Cranbury, NJ), was dissolved in saline to obtain doses of 50, 100, and 200 μg/kg/ml, and injected s.c. 5 min before each behavioral test. An equal volume of saline was administered to control animals[1]. |
| Alias | PT-141 Acetate |
| Molecular Weight | 1085.22 |
| Formula | C52H72N14O12 |
| Cas No. | 1607799-13-2 |
| Smiles | CC(O)=O.[H][C@]1(CCCCNC(=O)C[C@H](NC(=O)[C@H](CCCC)NC(C)=O)C(=O)N[C@@H](Cc2cnc[nH]2)C(=O)N[C@]([H])(Cc2ccccc2)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N1)C(O)=O |
| Relative Density. | no data available |
Storage & Solubility Information
| Storage | keep away from moisture,store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||
| Solubility Information | DMSO: 36 mg/mL (33.17 mM) | |||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||
DMSO
| ||||||||||||||||||||||||||
Calculator
In Vivo Formulation Calculator (Clear solution)
Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . A total of 10 animals were administered, and the formula you used is 5% 
DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
Dose Conversion
You can also refer to dose conversion for different animals. More Dose Conversion
Tech Support
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc
Keywords
Preview
Related Tags: buy Bremelanotide Acetate | purchase Bremelanotide Acetate | Bremelanotide Acetate cost | order Bremelanotide Acetate | Bremelanotide Acetate chemical structure | Bremelanotide Acetate in vivo | Bremelanotide Acetate formula | Bremelanotide Acetate molecular weight
- TOP
Feedback
Hello! How can I help you today? 
Copyright © 2015-2024 TargetMol Chemicals Inc. All Rights Reserved.