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PROTAC B-Raf degrader 1
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PROTAC B-Raf degrader 1
Catalog No. T12556Cas No. 2364367-27-9
PROTAC B-Raf degrader 1 is a proteolysis targeting chimera (PROTAC) for the degradation of B-Raf,PROTAC B-Raf degrader 1 With anti-cancer activity.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 5 mg | $431 | Backorder | |
| 10 mg | $689 | Backorder | |
| 50 mg | Inquiry | Backorder | |
| 100 mg | Inquiry | Backorder |
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CitedProduct Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | PROTAC B-Raf degrader 1 is a proteolysis targeting chimera (PROTAC) for the degradation of B-Raf,PROTAC B-Raf degrader 1 With anti-cancer activity. |
| In vitro | PROTAC B-Raf degrader 1 towards MCF-7, MDA-MB-231, HepG2, LO2 and B16 cells with IC50 values of 2.7 μM, 21.21 μM, 18.70 μM, 41.11μM and 22.68 μM, respectively[1]. |
| Molecular Weight | 763.77 |
| Formula | C36H37N5O12S |
| Cas No. | 2364367-27-9 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | |||||||||||||||||||||||||
| Solubility Information | DMSO: 25 mg/mL (32.73 mM), Sonication is recommended. | |||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||
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