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ST3932

ST3932
ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively).
Catalog No. T13008Cas No. 1246018-21-2

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ST3932

Catalog No. T13008Cas No. 1246018-21-2

ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively).
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Pack SizePriceAvailabilityQuantity
25 mg$1,6706-8 weeks
50 mg$2,1806-8 weeks
100 mg$2,8006-8 weeks
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Product Introduction

Bioactivity
Description
ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively).
Targets&IC50
A1 receptor:33 nM (ki), A2A receptor:ki: 8 nM
In vitro
ST3932 is a ST1535 metabolite, acts as an adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively). ST3932 inhibits agonist-induced cAMP accumulation(IC50 : 450 nM).
In vivo
In mice, Haloperidol-induced catalepsy antagonized by ST3932 (10, 20, 40 mg/kg, p.o.), and increases motor activity . ST3932 (20, 40 mg/kg, i.p.) significantly increases the number of contralateral turns induced by l-DOPA in rats.
Chemical Properties
Molecular Weight288.31
FormulaC12H16N8O
Cas No.1246018-21-2
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

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