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Taprenepag isopropyl

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Catalog No. T16988Cas No. 1005549-94-9
Alias PF-04217329

Taprenepag isopropyl is a highly selective agonist of the EP2 receptor.

Taprenepag isopropyl

Taprenepag isopropyl

😃Good
Catalog No. T16988Alias PF-04217329Cas No. 1005549-94-9
Taprenepag isopropyl is a highly selective agonist of the EP2 receptor.
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2 mg$485 days
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Product Introduction

Bioactivity
Description
Taprenepag isopropyl is a highly selective agonist of the EP2 receptor.
In vivo
Intraocular pressure (IOP) typically stays within normal limits in the left eye treated with a vehicle solution, while the right eye, dosed with Taprenepag isopropyl, shows a reduction in IOP across all dosage groups. Notably, in the high-dose group, IOP decreases to levels below measurable thresholds (<4mm Hg) on Days 22 and 29. Administration of Taprenepag isopropyl, regardless of the dose, does not result in clinical signs, body weight changes, or ocular findings in the animals receiving the lowest dose (0.75 mg/day) [1].
AliasPF-04217329
Chemical Properties
Molecular Weight520.6
FormulaC27H28N4O5S
Cas No.1005549-94-9
Relative Density.1.26 g/cm3 (Predicted)
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

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Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
1 Enter information below:
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2 Enter the in vivo formulation:
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Dose Conversion

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