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αvβ1 integrin-IN-1
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αvβ1 integrin-IN-1
Catalog No. T13473Cas No. 1689540-62-2
αvβ1 integrin-IN-1 is a potent and selective inhibitor of αvβ1 integrin (IC50 of 0.63 nM) with antifibrotic effects.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $129 | In Stock | |
| 5 mg | $315 | In Stock | |
| 10 mg | $495 | In Stock | |
| 25 mg | $791 | In Stock | |
| 50 mg | $1,120 | In Stock | |
| 100 mg | $1,490 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $466 | In Stock |
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Product Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | αvβ1 integrin-IN-1 is a potent and selective inhibitor of αvβ1 integrin (IC50 of 0.63 nM) with antifibrotic effects. |
| In vitro | In a murine model of liver and lung fibrosis, the administration of αvβ1 integrin-IN-1 leads to a significant reduction in the expression of fibrotic markers.[1] |
| Molecular Weight | 558.65 |
| Formula | C26H34N6O6S |
| Cas No. | 1689540-62-2 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | |||||||||||||||
| Solubility Information | DMSO: 5.59 mg/mL (10 mM)  | |||||||||||||||
Solution Preparation Table | ||||||||||||||||
DMSO
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