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Fidexaban
🥰Excellent
Catalog No. T27318Cas No. 183305-24-0
Alias ZK-807834, PD-200022, CI-1031, CI1031, BX-807834, BX807834
Fidexaban (CI1031) is a novel, potent, selective and orally active factor Xa inhibitor that has demonstrated antithrombotic activity in a variety of assays
Fidexaban
🥰Excellent
Purity: 99.42%
Catalog No. T27318Alias ZK-807834, PD-200022, CI-1031, CI1031, BX-807834, BX807834Cas No. 183305-24-0
Fidexaban (CI1031) is a novel, potent, selective and orally active factor Xa inhibitor that has demonstrated antithrombotic activity in a variety of assays
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | 135 € | In Stock | |
| 5 mg | 342 € | In Stock | |
| 10 mg | 503 € | In Stock | |
| 25 mg | 816 € | In Stock | |
| 50 mg | 1.121 € | In Stock | |
| 100 mg | 1.510 € | In Stock |
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Purity:99.42%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Fidexaban (CI1031) is a novel, potent, selective and orally active factor Xa inhibitor that has demonstrated antithrombotic activity in a variety of assays |
| Targets&IC50 | FXa (human):0.11 nM(Ki) |
| In vitro | Fidexaban (ZK-807834) is a novel, synthetic factor Xa (FXa) inhibitor with a Ki of 0.11 nM against human FXa. In human plasma in vitro, Fidexaban doubled PT and aPTT at 0.23 and 0.49 microM, respectively. Ex vivo plasma anti-FXa activity was also well correlated with plasma concentration of Fidexaban and with PT (r = 0.96 and 0.98, respectively).[2] |
| Alias | ZK-807834, PD-200022, CI-1031, CI1031, BX-807834, BX807834 |
| Molecular Weight | 526.49 |
| Formula | C25H24F2N6O5 |
| Cas No. | 183305-24-0 |
| Smiles | O(C1=C(F)C(N(CC(O)=O)C)=C(F)C(OC2=CC(=CC=C2)C=3N(C)CCN3)=N1)C4=CC(C(=N)N)=CC=C4O |
| Relative Density. | 1.31g/cm3 |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
| Solubility Information | DMSO: < 1 mg/mL (insoluble）  |
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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