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(Rac)-Managlinat dialanetil
(Rac)-Managlinat dialanetil ((Rac)-MB06322) is the racemate of Managlinat dialanetil, an orally available and potent inhibitor of fructose 1,6-bisphosphatase (FBPase) used in research 2 type diabetes.
Catalog No. T16009Cas No. 347870-26-2
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(Rac)-Managlinat dialanetil
Catalog No. T16009Cas No. 347870-26-2
(Rac)-Managlinat dialanetil ((Rac)-MB06322) is the racemate of Managlinat dialanetil, an orally available and potent inhibitor of fructose 1,6-bisphosphatase (FBPase) used in research 2 type diabetes.
With extensive experience in compound synthesis, we can provide rapid custom synthesis services for this product according to your research needs. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 25 mg | $1,970 | 6-8 weeks | |
| 50 mg | $2,580 | 6-8 weeks | |
| 100 mg | $3,400 | 6-8 weeks |
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Product Introduction
Bioactivity
Chemical Properties
| Description | (Rac)-Managlinat dialanetil ((Rac)-MB06322) is the racemate of Managlinat dialanetil, an orally available and potent inhibitor of fructose 1,6-bisphosphatase (FBPase) used in research 2 type diabetes. |
| In vivo | After oral administration, in Zucker diabetic fatty (ZDF) rats, Managlinat dialanetil dose-dependently inhibits GNG as well as lower basal and postprandial blood glucose levels[1]. |
| Alias | CS-917, (Rac)-MB06322, MB06322, (Rac)-CS-917 |
| Molecular Weight | 500.55 |
| Formula | C21H33N4O6PS |
| Cas No. | 347870-26-2 |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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