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A2B receptor antagonist 2
Catalog No. T37793Cas No. 784-90-7
Alias A2B receptor antagonist 2
A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).
A2B receptor antagonist 2
Catalog No. T37793Alias A2B receptor antagonist 2Cas No. 784-90-7
A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 10 mg | $38 | 1-2 weeks |
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Product Introduction
Bioactivity
Chemical Properties
| Description | A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B). |
| Targets&IC50 | A2A (rat):6.8 μM (Ki), A2B (human):3.44 μM (Ki), A1 (rat):2.30 μM (Ki) |
| Alias | A2B receptor antagonist 2 |
| Molecular Weight | 229.28 |
| Formula | C12H15N5 |
| Cas No. | 784-90-7 |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 2 mg/mL (8.72 mM), Sonication and heating to 60℃ are recommended. Methanol: 5 mg/mL (21.81 mM), Sonication and heating to 60℃ are recommended. | ||||||||||||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||||||||||||
DMSO/Methanol
Methanol
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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