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AZD-1897
🥰Excellent
Catalog No. T71242Cas No. 1204181-93-0
Alias AZD1897
AZD-1897 is a highly efficient ATP-competitive pan-PIM inhibitor with anticancer and antileukemic activity, inhibiting PIM1, PIM2, and PIM3, which can be used to study multiple myeloma.
AZD-1897
🥰Excellent
Purity: 99.49%
Catalog No. T71242Alias AZD1897Cas No. 1204181-93-0
AZD-1897 is a highly efficient ATP-competitive pan-PIM inhibitor with anticancer and antileukemic activity, inhibiting PIM1, PIM2, and PIM3, which can be used to study multiple myeloma.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $81 | In Stock | |
| 5 mg | $196 | In Stock | |
| 10 mg | $322 | In Stock | |
| 25 mg | $526 | In Stock | |
| 50 mg | $738 | In Stock | |
| 100 mg | $998 | In Stock | |
| 200 mg | $1,330 | In Stock |
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Purity:99.49%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | AZD-1897 is a highly efficient ATP-competitive pan-PIM inhibitor with anticancer and antileukemic activity, inhibiting PIM1, PIM2, and PIM3, which can be used to study multiple myeloma. |
| Targets&IC50 | PIM1/2/3:<3 nM |
| In vitro | AZD-1897 is a PIM1, PIM2, and PIM3 inhibitor with IC50 values of less than 3 nM. [1] |
| Alias | AZD1897 |
| Molecular Weight | 361.46 |
| Formula | C18H23N3O3S |
| Cas No. | 1204181-93-0 |
| Smiles | C(\C1=C(C(OC(C)C)=CC=C1)N2C[C@H](N)CCC2)=C/3\SC(=O)NC3=O |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||
| Solubility Information | DMSO: 16 mg/mL (44.26 mM), when pH is adjusted to 2 with HCL.Sonication and heating are recommended. | |||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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