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BAY 73-1449 is a potent and selective antagonist of the prostacyclin receptor (IC50 < 0.1 nM).
Pack Size | Price | Availability | Quantity |
---|---|---|---|
1 mg | $53 | In Stock | |
2 mg | $75 | In Stock | |
5 mg | $119 | In Stock | |
10 mg | $197 | In Stock | |
25 mg | $341 | In Stock | |
50 mg | $490 | In Stock | |
100 mg | $653 | In Stock | |
200 mg | $879 | In Stock | |
1 mL x 10 mM (in DMSO) | $136 | In Stock |
Description | BAY 73-1449 is a potent and selective antagonist of the prostacyclin receptor (IC50 < 0.1 nM). |
Targets&IC50 | Prostacyclin receptor:<0.1 nM |
In vivo | In male Wistar rats, BAY 73-1449 (0.1-1 mg/kg; i.v.) significantly reduced splenic shunt vessel outflow without affecting mesenteric inflow[1]. BAY 73-1449 (1-5 mg/kg; s.c.) has no effects on portal pressures and the degree of porto-systemic shunting in rats[1]. |
Alias | BAY73-1449, BAY-73-1449 |
Molecular Weight | 425.48 |
Formula | C26H23N3O3 |
Cas No. | 693790-96-4 |
Smiles | OC(=O)[C@@H](Cc1ccccc1)Nc1cc(ncn1)-c1ccc(OCc2ccccc2)cc1 |
Relative Density. | 1.273 g/cm3 (Predicted) |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
Solubility Information | DMSO: 55 mg/ml (129.27 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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