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CB1/2 agonist 3
Catalog No. T61736Cas No. 2772655-86-2
CB1/2 agonist 3 is a competitive and potent CB1/CB2 agonist with high affinity for hCB1 and hCB2 and can be used to study neurological disorders.
CB1/2 agonist 3
Catalog No. T61736Cas No. 2772655-86-2
CB1/2 agonist 3 is a competitive and potent CB1/CB2 agonist with high affinity for hCB1 and hCB2 and can be used to study neurological disorders.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $35 | In Stock | |
| 5 mg | $81 | In Stock | |
| 10 mg | $133 | In Stock | |
| 25 mg | $218 | In Stock | |
| 50 mg | $325 | In Stock | |
| 100 mg | $483 | In Stock |
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | CB1/2 agonist 3 is a competitive and potent CB1/CB2 agonist with high affinity for hCB1 and hCB2 and can be used to study neurological disorders. |
| Targets&IC50 | CB2-CHO cells (human):1.28 nM (EC50), CP-55940:78.17 nM (Kb), CB1-CHO cells (human):30.99 nM (EC50) |
| In vitro | CB1/2 agonist 3 partially induced the binding of [35S]GTPγS to hCB1-CHO cell membranes with an EC50=30.99 nM and slightly inhibited the binding of [35S]GTPγS to hCB2-CHO cell membranes with an average EC50=1.28 nM. CB1/2 agonist 3, after treatment for 1 hour at a concentration of 1 μM , antagonized the CB1/CB2 agonist CP-55940 with Kb=78.17 nM. [1] |
| Molecular Weight | 387.6 |
| Formula | C25H41NO2 |
| Cas No. | 2772655-86-2 |
Storage & Solubility Information
| Storage | keep away from moisture | Shipping with blue ice. | |||||||||||||||||||||||||
| Solubility Information | DMSO: 8 mg/mL(20.64 mM), Sonication is recommended. | |||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||
DMSO
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DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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