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CB2 receptor agonist 2
🥰Excellent
Catalog No. T22009Cas No. 1314230-75-5
Alias ZINC72105556, 4-Quinolone-3-Carboxamide Furan CB2 Agonist
CB2 receptor agonist 2 (ZINC72105556) is a potent and selective agonist for the CB2 (cannabinoid type 2) receptor, Ki = 8.5 nM. CB2 receptor agonist 2 has high affinity and selectivity for CB2.
CB2 receptor agonist 2
🥰Excellent
Purity: 98.07%
Catalog No. T22009Alias ZINC72105556, 4-Quinolone-3-Carboxamide Furan CB2 AgonistCas No. 1314230-75-5
CB2 receptor agonist 2 (ZINC72105556) is a potent and selective agonist for the CB2 (cannabinoid type 2) receptor, Ki = 8.5 nM. CB2 receptor agonist 2 has high affinity and selectivity for CB2.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $118 | In Stock | |
| 2 mg | $178 | In Stock | |
| 5 mg | $281 | In Stock | |
| 10 mg | $412 | In Stock | |
| 25 mg | $648 | In Stock | |
| 50 mg | $870 | In Stock | |
| 100 mg | $1,170 | In Stock |
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Purity:98.07%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | CB2 receptor agonist 2 (ZINC72105556) is a potent and selective agonist for the CB2 (cannabinoid type 2) receptor, Ki = 8.5 nM. CB2 receptor agonist 2 has high affinity and selectivity for CB2. |
| In vitro | CB2 receptor agonist 2 (compound 4g) (1 μM, 72 hours) exhibits minimal to no cytotoxicity in Hep-G2 cells[1]. |
| In vivo | CB2 receptor agonist 2 (compound 4g) (1 and 3 mg/kg; 1 hour) is highly potent, showing maximal effect at 1 mg/kg, with antihyperalgesic effects that are effective in the first phase of the nocifensive response and are strongly reduced by AM630, a CB2-selective antagonist/inverse agonist [1]. |
| Alias | ZINC72105556, 4-Quinolone-3-Carboxamide Furan CB2 Agonist |
| Molecular Weight | 488.62 |
| Formula | C30H36N2O4 |
| Cas No. | 1314230-75-5 |
| Smiles | N(C(=O)C=1C(=O)C=2C(N(CCCCC)C1)=C(OC)C=C(C2)C3=CC=CO3)C45CC6CC(C4)CC(C5)C6 |
| Relative Density. | no data available |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||
| Solubility Information | DMSO: 3 mg/mL (6.1 mM) | |||||||||||||||
Solution Preparation Table | ||||||||||||||||
DMSO
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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