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CB2 receptor agonist 2

Catalog No. T22009Cas No. 1314230-75-5
Alias ZINC72105556, 4-Quinolone-3-Carboxamide Furan CB2 Agonist

CB2 receptor agonist 2 (ZINC72105556) is a potent and selective agonist for the CB2 (cannabinoid type 2) receptor, Ki = 8.5 nM. CB2 receptor agonist 2 has high affinity and selectivity for CB2.

CB2 receptor agonist 2

CB2 receptor agonist 2

Purity: 98.07%
Catalog No. T22009Alias ZINC72105556, 4-Quinolone-3-Carboxamide Furan CB2 AgonistCas No. 1314230-75-5
CB2 receptor agonist 2 (ZINC72105556) is a potent and selective agonist for the CB2 (cannabinoid type 2) receptor, Ki = 8.5 nM. CB2 receptor agonist 2 has high affinity and selectivity for CB2.
Pack SizePriceAvailabilityQuantity
1 mg$118In Stock
2 mg$178In Stock
5 mg$281In Stock
10 mg$412In Stock
25 mg$648In Stock
50 mg$870In Stock
100 mg$1,170In Stock
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Purity:98.07%
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Product Introduction

Bioactivity
Description
CB2 receptor agonist 2 (ZINC72105556) is a potent and selective agonist for the CB2 (cannabinoid type 2) receptor, Ki = 8.5 nM. CB2 receptor agonist 2 has high affinity and selectivity for CB2.
In vitro
CB2 receptor agonist 2 (compound 4g) (1 μM, 72 hours) exhibits minimal to no cytotoxicity in Hep-G2 cells[1].
In vivo
CB2 receptor agonist 2 (compound 4g) (1 and 3 mg/kg; 1 hour) is highly potent, showing maximal effect at 1 mg/kg, with antihyperalgesic effects that are effective in the first phase of the nocifensive response and are strongly reduced by AM630, a CB2-selective antagonist/inverse agonist [1].
AliasZINC72105556, 4-Quinolone-3-Carboxamide Furan CB2 Agonist
Chemical Properties
Molecular Weight488.62
FormulaC30H36N2O4
Cas No.1314230-75-5
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
DMSO: 3 mg/mL (6.1 mM)
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.0466 mL10.2329 mL20.4658 mL102.3290 mL
5 mM0.4093 mL2.0466 mL4.0932 mL20.4658 mL

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