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ERK2 IN-1
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Catalog No. T11228Cas No. 1093061-47-2
ERK2 IN-1, a selective ERK2 inhibitor, exhibits an IC50 of 7 nM.
ERK2 IN-1
😃Good
Catalog No. T11228Cas No. 1093061-47-2
ERK2 IN-1, a selective ERK2 inhibitor, exhibits an IC50 of 7 nM.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 25 mg | $2,270 | 10-14 weeks | |
| 50 mg | $2,980 | 10-14 weeks | |
| 100 mg | $4,000 | 10-14 weeks |
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Product Introduction
Bioactivity
Chemical Properties
| Description | ERK2 IN-1, a selective ERK2 inhibitor, exhibits an IC50 of 7 nM. |
| Targets&IC50 | ERK2:7 nM |
| In vitro | ERK1/2 IN-1 maintains good ERK enzymatic activity and cellular activity in BRAF/KRAS mutant wildtype cancer cell lines . |
| Molecular Weight | 647.76 |
| Formula | C36H34FN7O2S |
| Cas No. | 1093061-47-2 |
| Relative Density. | 1.41 g/cm3 (Predicted) |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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