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GALNON
Catalog No. T8456Cas No. 475115-35-6
Galnon is a galanin receptor agonist, improves intrinsic cortical bone tissue properties
GALNON
Catalog No. T8456Cas No. 475115-35-6
Galnon is a galanin receptor agonist, improves intrinsic cortical bone tissue properties
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 25 mg | $817 | 1-2 weeks |
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Product Introduction
Bioactivity
Chemical Properties
| Description | Galnon is a galanin receptor agonist, improves intrinsic cortical bone tissue properties |
| In vivo | Galnon has been characterized to inhibit seizures, decrease feeding behaviour, diminish physical signs of opiate withdrawal and to alleviate heat-hyperalgesic response to partial sciatic nerve injury[1]. Galnon, a GAL receptor agonist, may enhance osteoclastic bone resorption in OVX rats. Although galnon reduced bone volume, biomechanical testing revealed that bone of galnon-treated animals was mechanically superior per unit area. Taken together, galnon simultaneously improves the intrinsic quality of cortical bone whilst stimulating osteoclastic activity in the OVX rat model[2]. |
| Molecular Weight | 678.82 |
| Formula | C40H46N4O6 |
| Cas No. | 475115-35-6 |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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