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Search Result

Search Results for " anxiolytic "

Targets

GABA Receptor

199

Compounds

23

Natural Products

4

Recombinant Proteins

Cat No. Product Name Synonyms Targets
T23445 Anxiolytic/nonsedative agent-1 TCS 1205 GABA Receptor
Anxiolytic/nonsedative agent-1 (TCS 1205) is a potent and selective GABAA agonist. Anxiolytic/nonsedative agent-1 shows appreciable affinity for the BzR in bovine brain membranes with Kis of 14, 121, 239 nM for α1β2γ2, α...
T15275 Fenobam GluR
Fenobam shows inverse agonist activity which blocks the mGlu5 receptor basal activity(IC50: 84 nM). Fenobam has anxiolytic activity. Fenobam is a selective and non-competitive mGluR5 antagonist acting at an allosteric mo...
T9626 Cycloleucine NMDAR
Cycloleucine is an antagonist of NMDA receptor associated glycine receptor with a Ki of 600 μM. Cycloleucine is also a competitive inhibitor of S-adenosyl-methionine mediated methylation with anxiolytic and cytostatic ef...
T1292 Tiapride hydrochloride Dopamine Receptor
Tiapride is a selective blocker of D2/3 dopamine receptors in the brain. It is used in the therapy of various psychiatric and neurological disorders containing dyskinesia, negative symptoms of psychosis, alcohol withdraw...
T2599 Pirenperone 5-HT Receptor
Pirenperone is a putative 5-HT2 receptor antagonist with the central antiserotonergic and antidopaminergic action.
T34896 Tofisopam Emandaxin,Grandaxin Others
Tofisopam (Grandaxin) is a 2,3-benzodiazepine compound with anxiolytic activity that can be taken orally.
T4508 Glycyl-L-Histidyl-L-Lysine Others
Glycyl-L-histidyl-L-lysine is a liver cell growth factor and an asynthetic hepatotrophic agent that stimulates hepatic erythropoietic factor production.
T13318 VU0650786 GluR
VU0650786 is a selective and potent CNS penetrant negative allosteric modulator of metabotropic glutamate receptor subtype 3 (mGlu3 NAM) (IC50: 392 nM), with antidepressant and anxiolytic activity in rodents.
T27475 GSK356278 GSK-356278,GSK 356278 PDE
GSK356278 is an effective and selective inhibitor of phosphodiesterase 4 (PDE4), with pIC50s of 8.6, 8.8, and 8.7 for human PDE4A, PDE4B, and PDE4D, respectively. GSK356278 has anti-inflammatory, anxiolytic, and cognitio...
T19680 Zotepine Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor , Histamine Receptor
Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM, 3.3 nM, 7.3 nM, and 8 nM, respectively. Zotepine is a second...
T15286 Flindokalner BMS-204352 Potassium Channel
Flindokalner (BMS-204352) is a potassium channel modulator and a positive modulator of all neuronal Kv7 channel subtypes expressed in HEK293 cells. Flindokalner is a large conductance calcium-activated K channel (BKca) p...
T6022 LY404039 pomaglumetad Glucocorticoid Receptor , GluR
LY404039 (pomaglumetad) is an effective agonist of recombinant human mGlu2(Ki =149 nM)/mGlu3(Ki =92 nM).
T21995 XAP044 GluR
XAP044 is a mGlu7-selective antagonist which inhibits lateral amygdala long term potentiation (LTP) in brain slices from wild type mice with a half-maximal blockade at 88 nm[1].
T8004 SNAP 94847 hydrochloride GPR , Melanin-concentrating Hormone Receptor (MCHR)
SNAP 94847 hydrochloride is a melanin-concentrating hormonereceptor1 (MCHR1) antagonist(Ki= 2.2 nM)
T4176 Rac-BHFF (R,S)-BHFF GABA Receptor
rac-BHFF ((R,S)-BHFF) is potent and selective GABA B receptor positive allosteric modulator that increases the potency and efficacy of GABA ( > 15-fold and > 149% respectively). It exhibits anxiolytic activity in vivo an...
T8887 2'MeO6MF GABA Receptor
2'MeO6MF is a brain-penetrant positive allosteric modulator at α2β1γ2L and all α1-containing GABAA receptors.It offers neuroprotection and improved functional recovery and dampens the stroke-induced inflammatory response...
T8357 SB-200646 5-HT Receptor
SB-200646 is a selective and potent antagonist of 5-HT2B/5-HT2C receptor
TQ0311 GSK163090 Dopamine Receptor , 5-HT Receptor
GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3).
T11393 GET73 Gamma hydroxybutyric acid analogue,GET 73 GluR
GET73 (Gamma hydroxybutyric acid analogue) is an negative allosteric modulator of mGluR5. GET73 is a naturally occurring neurotransmitter. GET73 has anti-alcohol and anxiolytic properties.
T0162 Quetiapine ICI204636,Quetiapin Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor , AChR , Histamine Receptor
Quetiapine (ICI204636) is used for the therapy of schizophrenia, and for the treatment of acute manic episodes associated with bipolar I disorder. The mechanism of quetiapine' action is thought by mediated through antago...
T19916 TRIM 1-(2-Trifluoromethylphenyl)imidazole NOS
TRIM (1-(2-Trifluoromethylphenyl)imidazole) is an inhibitor of nNOS.
T13690 Etifoxine hydrochloride HOE 36-801 hydrochloride GABA Receptor
Etifoxine hydrochloride (HOE 36-801 hydrochloride) is an anxiolytic and anticonvulsant drug. Unlike benzodiazepines, Etifoxine hydrochloride appears to produce its anxiolytic effects by binding to β2 and β3 subunits of t...
TP2206 [Leu31,Pro34]-Neuropeptide Y (porcine) Neuropeptide Y Receptor
High affinity neuropeptide Y Y1 receptor agonist
T6241 Quetiapine hemifumarate Quetiapine Fumarate,ICI-204636 Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor
Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar II depression, bipolar I depression.
T27835 Lin281632 Lin-28 1632,Lin-281632,Lin 281632,Lin28 1632,Lin 28 163
Lin28 1632 is an inhibitor of RNA binding protein Lin28. It promotes mESC differentiation. Lin281632 is also bromodomain inhibitor.
T15022 CVT-10216 Dehydrogenase
CVT-10216 is a Potent and selective, reversible inhibitor of aldehyde dehydrogenase 2 (ALDH2) (IC50: 29 nM). CVT-10216 also has inhibitory effect of ALDH-1 (IC50: 1.3 μM). CVT-10216 can reduce excessive alcohol drinking...
T8456 GALNON Neuropeptide Y Receptor
Galnon is a galanin receptor agonist, improves intrinsic cortical bone tissue properties
T14204 6-Iodopravadoline AM630 Cannabinoid Receptor
6-Iodopravadoline (AM630) is an antagonist of CB2 (Ki: 31.2 nM). And it shows 165-fold selectivity more than CB1 receptors.
T5135 Flupentixol dihydrochloride Fupentixol Dihydrochloride,Flupenthixol dihydrochloride,(E/Z)-Flupentixol Dihydrochloride Dopamine Receptor
Flupentixol dihydrochloride is used in therapy of schizophrenia as well as in anxiolytic and depressive disorders.
T6888 Methylene Blue methylthioninium chloride,CI-52015,Tetramethylthionine chloride,Basic Blue 9 Guanylate cyclase , Microtubule Associated , NO Synthase , Parasite , Monoamine Oxidase
Methylene Blue (Tetramethylthionine chloride) (IC50 of 1.9 μM) inhibits tau filament formation. And it inhibits soluble guanylyl cyclase. It is also used as a dye in chromoendoscopy.
T5406 SNAP 94847 SNAP-94847 GPR , Melanin-concentrating Hormone Receptor (MCHR)
SNAP 94847 (SNAP-94847) is a selective and competitive MCH1 receptor (MCH1-R) antagonist (Ki: 2.2 nM). It has anxiolytic and antidepressant activity and reduces food intake in mice.
T0006 Methylene Blue trihydrate Methylthionine chloride,Basic blue 9,Methylene Blue Guanylate cyclase , Microtubule Associated , NO Synthase , Parasite , Monoamine Oxidase
Methylene Blue trihydrate (Basic blue 9) is a compound consisting of dark green crystals or crystalline powder, having a bronze-like luster. Solutions in water or alcohol have a deep blue color. Methylene Blue trihydrate...
T28662 Saripidem SL-850274,SL-85.0274,SL850274,SL85.0274 Others
Saripidem (SL-85.0274) is a compound with anxiolytic activity.
T1864 Fabomotizole Obenoxazine,CM346 Others
Fabomotizole (Obenoxazine) is an anxiolytic drug; produces anxiolytic and neuroprotective effects without any sedative or muscle relaxant actions.
T61816 EMD 56551
EMD 56551 is a powerful and specific agonist of the 5-HT1A receptor, demonstrating significant anxiolytic properties [1].
T28303 Pazinaclone A-77000,DN-2327,DN2327,DN 2327,A 77000,A77000 GABA Receptor
Pazinaclone is a non-benzodiazepine (GABAA) partial agonist with sedative and anxiolytic activity.
T23007 MM 77 dihydrochloride FITC-Dextran (60842-46-8 MW 4000) 5-HT Receptor
MM 77 dihydrochloride is an effecitve 5-HT1A receptor postsynaptic antagonist with anxiolytic-like activity.
T4688 Pipequaline hydrochloride PK-8165 hydrochloride GABA Receptor
Pipequaline hydrochloride (PK-8165 hydrochloride) is an anticonflict & anticonvulsant quinoline derivative. It is an anxiolytic drug that was never marketed. It possesses a novel chemical structure that is not closely re...
T12847 SB-616234-A SB-616234A 5-HT Receptor
SB-616234A is a selective and orally bioavailable antagonist of 5-HT1B receptor, with anxiolytic and antidepressant activity.
T20515L Selank Acetate（129954-34-3，free） Others
Selank Acetate is a typical anxiolytic producing no side effects.
T60195 Acetophenazine Others
Acetophenazine is an anxiolytic compound that is used in the study of depression.
T7107 δ-Sleep Inducing Peptide DSIP,Delta-Sleep Inducing Peptide Antioxidant
δ-Sleep Inducing Peptide (DSIP) is a neuropeptide, with antioxidant and anxiolytic properties.
T32845 Lofendazam Bu 1014
Lofendazam (Bu 1014) is a benzodiazepine derivative that has sedative and anxiolytic effects.
T4093 Fabomotizole hydrochloride Afobazole hydrochloride,CM346 hydrochloride MAO
Fabomotizole hydrochloride (CM346 hydrochloride), an anxiolytic drug, produces anxiolytic and neuroprotective effects. The mechanism of Afobazole remains poorly defined, however, with GABAergic, NGF, and BDNF release pro...
T27186 Divaplon RU-32698,RU32698,RU 32698 GABA Receptor
Divaplon is a GABA receptor agonist (IC50: 0.056 µM) that displays non-sedating anxiolytic behavioral characteristics in a rat model of anxiety.
T27001 CGS8216 CGS 8216,CGS-8216 Others
CGS8216 is a benzodiazepine receptor antagonist that shows analgesic activity at high doses.CGS8216 has anxiolytic activity and may be used to study immune system disorders.
T12841 SB-224289 hydrochloride SB-224289A 5-HT Receptor
SB-224289 hydrochloride (SB-224289A) is a selective antagonist of 5-HT1B receptor, with anxiolytic effect.
T5474 D159687 D 159687 PDE
D159687 is a selective PDE4D inhibitor,had a procognitive profile as it improved memory in the novel object recognition test but had no antidepressant or anxiolytic benefit.
T27262 Enciprazine WY-48624,D-3112,WY48624,WY 48624,D 3112,D3112 5-HT Receptor
Enciprazine (D-3112) has anxiolytic activity with high affinity for 5-HT1A receptor and ADRA1, which can be used for the treatment of anxiety disorders and can be used to study depression.
T12441 Phenelzine sulfate Monoamine Oxidase
Phenelzine sulfate is a non-selective and irreversible inhibitor of monoamine oxidase (MAOI), and with antidepressant and anxiolytic.

Compounds

Anxiolytic/nonsedative agent-1
T23445
Synonym: TCS 1205
Target: GABA Receptor
Fenobam
T15275
Synonym:
Target: GluR
Cycloleucine
T9626
Synonym:
Target: NMDAR
Tiapride hydrochloride
T1292
Synonym:
Target: Dopamine Receptor
Pirenperone
T2599
Synonym:
Target: 5-HT Receptor
Tofisopam
T34896
Synonym: Emandaxin,Grandaxin
Target: Others
Glycyl-L-Histidyl-L-Lysine
T4508
Synonym:
Target: Others
VU0650786
T13318
Synonym:
Target: GluR
GSK356278
T27475
Synonym: GSK-356278,GSK 356278
Target: PDE
Zotepine
T19680
Synonym:
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, Histamine Receptor
Flindokalner
T15286
Synonym: BMS-204352
Target: Potassium Channel
LY404039
T6022
Synonym: pomaglumetad
Target: Glucocorticoid Receptor, GluR
XAP044
T21995
Synonym:
Target: GluR
SNAP 94847 hydrochloride
T8004
Synonym:
Target: GPR, Melanin-concentrating Hormone Receptor (MCHR)
rac-BHFF
T4176
Synonym: (R,S)-BHFF
Target: GABA Receptor
2'MeO6MF
T8887
Synonym:
Target: GABA Receptor
SB-200646
T8357
Synonym:
Target: 5-HT Receptor
GSK163090
TQ0311
Synonym:
Target: Dopamine Receptor, 5-HT Receptor
GET73
T11393
Synonym: Gamma hydroxybutyric acid analogue,GET 73
Target: GluR
Quetiapine
T0162
Synonym: ICI204636,Quetiapin
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, AChR, Histamine Receptor
TRIM
T19916
Synonym: 1-(2-Trifluoromethylphenyl)imidazole
Target: NOS
Etifoxine hydrochloride
T13690
Synonym: HOE 36-801 hydrochloride
Target: GABA Receptor
[Leu31,Pro34]-Neuropeptide Y (porcine)
TP2206
Synonym:
Target: Neuropeptide Y Receptor
Quetiapine hemifumarate
T6241
Synonym: Quetiapine Fumarate,ICI-204636
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor
Lin281632
T27835
Synonym: Lin-28 1632,Lin-281632,Lin 281632,Lin28 1632,Lin 28 163
Target:
CVT-10216
T15022
Synonym:
Target: Dehydrogenase
GALNON
T8456
Synonym:
Target: Neuropeptide Y Receptor
6-Iodopravadoline
T14204
Synonym: AM630
Target: Cannabinoid Receptor
Flupentixol dihydrochloride
T5135
Synonym: Fupentixol Dihydrochloride,Flupenthixol dihydrochloride,(E/Z)-Flupentixol Dihydrochloride
Target: Dopamine Receptor
Methylene Blue
T6888
Synonym: methylthioninium chloride,CI-52015,Tetramethylthionine chloride,Basic Blue 9
Target: Guanylate cyclase, Microtubule Associated, NO Synthase, Parasite, Monoamine Oxidase
SNAP 94847
T5406
Synonym: SNAP-94847
Target: GPR, Melanin-concentrating Hormone Receptor (MCHR)
Methylene Blue trihydrate
T0006
Synonym: Methylthionine chloride,Basic blue 9,Methylene Blue
Target: Guanylate cyclase, Microtubule Associated, NO Synthase, Parasite, Monoamine Oxidase
Saripidem
T28662
Synonym: SL-850274,SL-85.0274,SL850274,SL85.0274
Target: Others
Fabomotizole
T1864
Synonym: Obenoxazine,CM346
Target: Others
EMD 56551
T61816
Synonym:
Target:
Pazinaclone
T28303
Synonym: A-77000,DN-2327,DN2327,DN 2327,A 77000,A77000
Target: GABA Receptor
MM 77 dihydrochloride
T23007
Synonym: FITC-Dextran (60842-46-8 MW 4000)
Target: 5-HT Receptor
Pipequaline hydrochloride
T4688
Synonym: PK-8165 hydrochloride
Target: GABA Receptor
SB-616234-A
T12847
Synonym: SB-616234A
Target: 5-HT Receptor
Selank Acetate（129954-34-3，free）
T20515L
Synonym:
Target: Others
Acetophenazine
T60195
Synonym:
Target: Others
δ-Sleep Inducing Peptide
T7107
Synonym: DSIP,Delta-Sleep Inducing Peptide
Target: Antioxidant
Lofendazam
T32845
Synonym: Bu 1014
Target:
Fabomotizole hydrochloride
T4093
Synonym: Afobazole hydrochloride,CM346 hydrochloride
Target: MAO
Divaplon
T27186
Synonym: RU-32698,RU32698,RU 32698
Target: GABA Receptor
CGS8216
T27001
Synonym: CGS 8216,CGS-8216
Target: Others
SB-224289 hydrochloride
T12841
Synonym: SB-224289A
Target: 5-HT Receptor
D159687
T5474
Synonym: D 159687
Target: PDE
Enciprazine
T27262
Synonym: WY-48624,D-3112,WY48624,WY 48624,D 3112,D3112
Target: 5-HT Receptor
Phenelzine sulfate
T12441
Synonym:
Target: Monoamine Oxidase
1 2 3 4
Cat No. Product Name Synonyms Targets
T3886 Rosavin Rosavidin P450
Rosavin (Rosavidin) has antidepressant and anxiolytic actions, helps balance all the neurotransmitters.
T5661 Methyl isoeugenol Others
methyl isoeugenol (MIE) is a natural food flavour that constitutes 93.7% of an essential oil from Pimenta pseudocaryophyllus leaf. The leaf extracts of this species are used as a calming agent. As a ubiquitous food addit...
T8014 Epoxylinalool 2-(2-Hydroxy-2-Propyl)-5-Methyl-5-Vinyltetrahydrofuran Others
Epoxylinalool (2-(2-Hydroxy-2-Propyl)-5-Methyl-5-Vinyltetrahydrofuran) is a naturally occurring monoterpene alcohol widely used in the production of perfumes and flavors.
T2719 Succinic acid Asuccin,Amber acid,1,2-Ethanedicarboxylic acid,Wormwood acid,Butanedioic acid,1,4-Butandioic Acid Endogenous Metabolite
Succinic acid (1,2-Ethanedicarboxylic acid) is a water-soluble, colorless crystal with an acid taste that is used as a chemical intermediate, in medicine, the manufacture of lacquers, and to make perfume esters. It is al...
T1045 Trimipramine maleate Surmontil maleate Dopamine Receptor , 5-HT Receptor , Antibacterial , Adrenergic Receptor , Norepinephrine , Histamine Receptor
Trimipramine maleate (Surmontil maleate) appears to inhibit serotonin transport and norepinephrine uptake by nerve terminals. This increases available norepinephrine or serotonin and prolongs its action. Trimipramine Mal...
T3748 Orcinol 5-Methylresorcinol,3,5-Dihydroxytoluene,5-Methylresorcin,3,5-ToluenediolOrcin,5-Methyl-1,3-benzenediol,Orcin Others
orcinol (5-Methylresorcin) is anxiolytic agent without sedative effect.
T4S0675 Polygalasaponin V Others
Polygalasaponin possesses evident anxiolytic and sedative-hypnotic activities and has a relatively safe dose range, which supports the use of Polygala tenuifolia root as an anxiolytic and sedative-hypnotic drug in folk m...
T4591 Dihydrokavain Marindinin,7,8-Dihydrokavain,7,8-Dihydrokawain Others
Dihydrokavain (Marindinin), a prominent kavalactone in the kava plant, significantly contributes to the plant's anxiolytic effects, as evidenced by a study conducted on chicks.
TN4114 Gardenin A ERK , LDL , MAPK , PKA , PKC
Gardenin A shows neurotrophic effects via activating MAPK/ERK, PKC, and PKA. Gardenin A exhibits antidepressant, anticonvulsant and anxiolytic effects.
TN1560 Dehydroeffusol 5-Ethenyl-1-Methylphenanthrene-2,7-Diol,Dehydro Effusol MMP , ERK , GPR , Others
Dehydroeffusol (Dehydro Effusol) possesses anti-cancer, anxiolytic and sedative properties. Dehydroeffusol inhibits gastric cancer cell growth and tumorigenicity by selectively inducing tumor-suppressive endoplasmic reti...
T2771 Orcinol glucoside Sakakin Antioxidant
Orcinol glucoside (Sakakin) (OG), an active constituent isolated from the rhizomes of Curculigo orchioides Gaertn, shows potent antioxidative and anxiolytic activities without sedative effects.
T4S1990 Carvacrol Karvakrol,O-Thymol,cymophenol Apoptosis , Others , Gamma-secretase , Endogenous Metabolite , Antifungal
1. Carvacrol (O-Thymol) presents anxiolytic effects. 2. 5-Isopropyl-2-methylphenol presents antinociceptive activity. 3. Carvacrol presents antidepressant effects, seems to be dependent on its interaction with the dopami...
T3S1319 (+)-Magnoflorine Escholin,Magnoflorine,Thalictrin,Escholine Others , Antifungal
(+)-Magnoflorine (Thalictrin) has sedative and anxiolytic effects, probably mediated by Magnoflorine through a GABAergic mechanism of action. Magnoflorine and Sinomenine have protective effects, are mediated by some mech...
T4S1999 Valepotriate Valtrate Apoptosis , HIV Protease
Valepotriate (Valtrate) fraction can have sedative effects and affect behavioral parameters related to recognition memory. Valepotriates, a new class of cytotoxic and antitumor agents, they are very potent cytotoxic agen...
T6S2227 Spinosin Flavoayamenin Others
1. Spinosin (Flavoayamenin) ameliorated memory impairment induced through AβO, the serotonergic neurotransmitter system, and these effects were regulated, in part, through neuroprotective activity via the anti-inflammato...
TN5166 Trans-Methylisoeugenol Parasite , GST
Trans-Methylisoeugenol is a compound with insecticidal activity isolated from Acorus calamus L. It is a natural food flavor. It is a natural food flavor with anxiolytic and antidepressant properties and moderately revers...
TCS0102 Pulegone (+)-Pulegone Calcium Channel , Endogenous Metabolite , TRP/TRPV Channel
1. Pulegone ((+)-Pulegone) has cytotoxicity followed by regenerative cell proliferation is the MOA for Pulegone-induced urothelial tumors in female rats. 2. Pulegone induces a verapamil-sensitive psychostimulant effect t...
TN1814 Juncusol Caspase , Antifection
Juncusol shows anxiolytic and sedative activities, it shows anxiolytic activity at dosages of 10 mg/kg; it can induce caspase-3-mediated cytotoxicity in HT22 cells. Juncusol has anti-microbial activity, it shows signific...
TN1678 Gelsevirine Others
Gelsevirine has anxiolytic activity, may be via the agonist action of glycine receptor in the brain.
TN4048 Exoticin Others
Exoticin shows antinociceptive and neuropharmacological activities, it could be considered as a suitable candidate for the development of analgesic and anxiolytic agents.
T72382 Dihydro-β-erythroidine
Dihydro-β-erythroidine, a competitive nicotinic receptor antagonist, effectively blocks the discriminative stimulus properties and inhibits the anxiolytic effects induced by nicotine.
TN5147 Tilifodiolide IL Receptor , TNF , GABA Receptor
Tilifodiolide exerts in vitro and in vivo anti-inflammatory activity and in vivo antinociceptive effects. Tilifodiolide exerted antidiarrheal activity by decreasing the intestinal fluid accumulation and vasorelaxant effe...
TN4322 Isopulegol ATPase , Potassium Channel , GABA Receptor
Isopulegol presents depressant- and anxiolytic-like effects, it also has anticonvulsant and bioprotective effects against PTZ-induced convulsions are possibly related to positive modulation of benzodiazepine-sensitive GA...

Natural Products

Rosavin
T3886
Synonym: Rosavidin
Target: P450
Methyl isoeugenol
T5661
Synonym:
Target: Others
Epoxylinalool
T8014
Synonym: 2-(2-Hydroxy-2-Propyl)-5-Methyl-5-Vinyltetrahydrofuran
Target: Others
Succinic acid
T2719
Synonym: Asuccin,Amber acid,1,2-Ethanedicarboxylic acid,Wormwood acid,Butanedioic acid,1,4-Butandioic Acid
Target: Endogenous Metabolite
Trimipramine maleate
T1045
Synonym: Surmontil maleate
Target: Dopamine Receptor, 5-HT Receptor, Antibacterial, Adrenergic Receptor, Norepinephrine, Histamine Receptor
orcinol
T3748
Synonym: 5-Methylresorcinol,3,5-Dihydroxytoluene,5-Methylresorcin,3,5-ToluenediolOrcin,5-Methyl-1,3-benzenediol,Orcin
Target: Others
Polygalasaponin V
T4S0675
Synonym:
Target: Others
Dihydrokavain
T4591
Synonym: Marindinin,7,8-Dihydrokavain,7,8-Dihydrokawain
Target: Others
Gardenin A
TN4114
Synonym:
Target: ERK, LDL, MAPK, PKA, PKC
Dehydroeffusol
TN1560
Synonym: 5-Ethenyl-1-Methylphenanthrene-2,7-Diol,Dehydro Effusol
Target: MMP, ERK, GPR, Others
Orcinol glucoside
T2771
Synonym: Sakakin
Target: Antioxidant
Carvacrol
T4S1990
Synonym: Karvakrol,O-Thymol,cymophenol
Target: Apoptosis, Others, Gamma-secretase, Endogenous Metabolite, Antifungal
(+)-Magnoflorine
T3S1319
Synonym: Escholin,Magnoflorine,Thalictrin,Escholine
Target: Others, Antifungal
Valepotriate
T4S1999
Synonym: Valtrate
Target: Apoptosis, HIV Protease
Spinosin
T6S2227
Synonym: Flavoayamenin
Target: Others
Trans-Methylisoeugenol
TN5166
Synonym:
Target: Parasite, GST
Pulegone
TCS0102
Synonym: (+)-Pulegone
Target: Calcium Channel, Endogenous Metabolite, TRP/TRPV Channel
Juncusol
TN1814
Synonym:
Target: Caspase, Antifection
Gelsevirine
TN1678
Synonym:
Target: Others
Exoticin
TN4048
Synonym:
Target: Others
Dihydro-β-erythroidine
T72382
Synonym:
Target:
Tilifodiolide
TN5147
Synonym:
Target: IL Receptor, TNF, GABA Receptor
Isopulegol
TN4322
Synonym:
Target: ATPase, Potassium Channel, GABA Receptor

Recombinant Proteins

Species：
Human (3)
Mouse (1)
Expression System：
E. coli (2)
HEK293 (1)
in vitro E. coli expression system (1)
Tag：
N-terminal 6xHis-KSI-tagged (2)
C-terminal hFc-tagged (1)
N-terminal 10xHis-tagged (1)
Cat No. Product Name Species Expression System
TMPH-00860 HTR1D Protein, Human, Recombinant (hFc) Human HEK293
G-protein coupled receptor for 5-hydroxytryptamine (serotonin). Also functions as a receptor for ergot alkaloid derivatives, various anxiolytic and antidepressant drugs and other psychoactive substances. Ligand binding c...
TMPH-00861 HTR1D Protein, Human, Recombinant (His & KSI) Human E. coli
G-protein coupled receptor for 5-hydroxytryptamine (serotonin). Also functions as a receptor for ergot alkaloid derivatives, various anxiolytic and antidepressant drugs and other psychoactive substances. Ligand binding c...
TMPH-00859 HTR1B Protein, Human, Recombinant (His) Human in vitro E. coli expression system
G-protein coupled receptor for 5-hydroxytryptamine (serotonin). Also functions as a receptor for ergot alkaloid derivatives, various anxiolytic and antidepressant drugs and other psychoactive substances, such as lysergic...
TMPH-02910 Somatostatin Protein, Mouse, Recombinant (His & KSI) Mouse E. coli
Inhibits the secretion of pituitary hormones, including that of growth hormone/somatotropin (GH1), PRL, ACTH, luteinizing hormone (LH) and TSH. Also impairs ghrelin- and GnRH-stimulated secretion of GH1 and LH; the inhib...
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