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Lesopitron HCl
🥰Excellent
Catalog No. T11839LCas No. 132449-88-8
Alias Lesopitron HCl(132449-89-9 Free base)
Lesopitron HCl is a 5-HT1A receptor agonist with anxiolytic effects that reverses dark avoidance behavior associated with cocaine withdrawal in mice.
Lesopitron HCl
🥰Excellent
Purity: 98.18%
Catalog No. T11839LAlias Lesopitron HCl(132449-89-9 Free base)Cas No. 132449-88-8
Lesopitron HCl is a 5-HT1A receptor agonist with anxiolytic effects that reverses dark avoidance behavior associated with cocaine withdrawal in mice.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $700 | In Stock | |
| 5 mg | $1,800 | In Stock |
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CitedSelect Batch
Purity:98.18%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Lesopitron HCl is a 5-HT1A receptor agonist with anxiolytic effects that reverses dark avoidance behavior associated with cocaine withdrawal in mice. |
| In vivo | E4424 (acute oral) increased adherent mucus levels by 12%, 11%, and 13%, relative to controls. Chronic E4424 significantly increased gastric mucus relative to controls (69% increase). E4424 has potent anti-gastric secretory and antiulcer effects.[1] |
| Alias | Lesopitron HCl(132449-89-9 Free base) |
| Molecular Weight | 357.28 |
| Formula | C15H22Cl2N6 |
| Cas No. | 132449-88-8 |
| Smiles | Cl.ClC=1C=NN(C1)CCCCN2CCN(C3=NC=CC=N3)CC2 |
| Relative Density. | no data available |
Storage & Solubility Information
| Storage | store at low temperature | Shipping with blue ice. | ||||||||||||||||||||
| Solubility Information | DMSO: 4.8 mg/mL (13.43 mM)  | ||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||
DMSO
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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