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Cell Cycle/Checkpoint MetabolismATP Citrate Lyase
(11)
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Serine/threonin kinase
Serine threonine kinase belongs to protein kinase, which can phosphorylate the OH group of serine or threonine residues. Serine threonine kinases contain Rho kinase, Aurora kinase, AMP kinase, RAF kinase, Polo like kinase, PIM kinase, ATM kinase and other kinases. The cAMP/cGMP, Ca2+/calmodulin and diacylglycerol and multiple chenmical signals can regulate the activity of serine threonine kinases.
- LP-935509T157811454555-29-3LP-935509 is highly brain-penetrant and reverses fully established pain behavior following the SNL procedure. LP-935509 is also an effective inhibitor of BIKE (IC50=14 nM) and a modest inhibitor of GAK (IC50=320 nM). LP-935509 is a selective, ATP-competit
- $33
SizeQTY
- (+)-Isocorydine hydrochlorideT429113552-72-2(+)-Isocorydine hydrochloride (Isocorydine HCl) is a eukaryote protein kinases Inhibitor.
- $37
SizeQTY - BMT-124110 FormateT10572L In houseBMT-124110 Formate is a selective AAK1 inhibitor (IC50: 0.9 nM) with anti-injury sensory activity.BMT-124110 Formate inhibits the BMP-2-inducible protein kinase BIKE with an IC50: 17 nM.BMT-124110 Formate inhibits the cell-cycle protein G-related BMT-124110 Formate inhibits the cell cycle protein G-associated kinase GAK with an IC50:99 nM.
- $195
SizeQTY
- FasudilT1606103745-39-7Fasudil (HA-1077) is a potent inhibitor of ROCK1, PKA, PKC, and MLCK.
- $33
SizeQTY - MLCK inhibitor peptide 18 acetateTP1890L1MLCK inhibitor peptide 18 acetate is a selective competitive inhibitor of myosin light chain kinase (IC50 = 50 nM). Displays 4000-fold selectivity over CaM kinase II and does not inhibit PKA. Cell permeable.
- $47
SizeQTY
Cited - N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamineT92561071135-06-2N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine is a novel 2,6-naphthyridine identified by high throughput screen (HTS) as a dual protein kinase C/D (PKC/PKD) inhibitor[1].
- $148
SizeQTY - HTH-01-091T241522000209-42-5In houseHTH-01-091 is a potent and selective maternal embryonic leucine zipper kinase (MELK) inhibitor (IC50: 10.5 nM).HTH-01-091 inhibits PIM1/2/3, RIPK2, DYRK3, smMLCK and CLK2. HTH-01-091 can be used to study breast cancer.
- $296
SizeQTY - WortmanninT628319545-26-7Wortmannin (SL-2052) is a PI3K inhibitor (IC50=3 nM) that is covalent and irreversible. Wortmannin is also an inhibitor of PlK1 and PlK3 (IC50=5.8/48 nM) that blocks autophagy.
- $32
SizeQTY Cited - ML-7 hydrochlorideT3050110448-33-4ML-7 hydrochloride (ML-7 HCl) is a cell-permeable, reversible, effective, ATP-competitive, and specific inhibitor of myosin light chain kinase (Ki: 300 nM); also inhibits smooth-muscle myosin light chain kinase, PKA, and PKC.
- $42
SizeQTY Cited - Camostat mesylateT239159721-29-8Camostat mesylate (FOY-S980) is a trypsin-like protease inhibitor and inhibits airway epithelial sodium channel (ENaC) function.
- $43
SizeQTY Cited - Fasudil hydrochlorideT3060105628-07-7Fasudil hydrochloride (HA-1077) is a potent inhibitor of ROCK1, PKA, PKC, and MLCK with Ki of 0.33 μM, 1.0 μM, 9.3 μM and 55 μM, respectively.
- $35
SizeQTY Cited - Nafamostat mesylateT239282956-11-4Nafamostat mesylate (FUT-175), a synthetic serine protease inhibitor, has been used for the treatment of allergic disorders such as asthma, allergic rhinitis and atopic dermatitis.
- $39
SizeQTY Cited - PiceatannolT061010083-24-6Piceatannol (Astringenin) is an anti-inflammatory, immunomodulatory and antiproliferative agent. It inhibits p56lck and syk protein tyrosine kinases and inhibits NF-κB activation and gene expression of TNF-induced. It is synthetic from the conversion of resveratrol by cytochrome P450 1B1.
- $39
SizeQTY Cited - CID 2011756T1863638156-11-3CID 2011756 is an ATP-competitive and specific PKD1 inhibitor.
- $39
SizeQTY - GAK inhibitor 49T8535319492-82-5GAK inhibitor 49 is a highly selective and ATP-competitive cyclin G associated kinase (GAK) inhibitor (IC50: 56 nM; Ki: 0.54 nM ).
- $87
SizeQTY - TAO Kinase inhibitor 2T77501850467-77-5TAO Kinase inhibitor 2 is a TAO kinase inhibitor with an IC50 of 50-500 nM. TAO Kinase inhibitor 2 inhibits KIAA1361 and JIK with IC50s of 50-500 nM.
- $30
SizeQTY - SRPKIN-1T169312089226-94-6SRPKIN-1 is a covalent and irreversible inhibitor of SRPK1/2 (IC50s: 35.6 and 98 nM, respectively).
- $297
SizeQTY - 1-NM-PP1T2153221244-14-01-NM-PP1 (PP1 Analog II) is a cell-permeable PP1 analog that acts as a potent and selective inhibitor of mutant kinases over their wild-type progenitors.
- $43
SizeQTY - CRT0066101 dihydrochloride(956121-30-5 free base)T8957L2308510-39-4CRT0066101 dihydrochloride is an inhibitor of PKD.
- $34
SizeQTY - IPR-803T11666892243-35-5IPR-803 is an effective inhibitor of the uPAR·uPA protein-protein interaction (PPI) with anti-tumor activity. IPR-803 binds directly to uPAR with a Ki of 0.2 μM.
- $84
SizeQTY - R-IMPPT40582133832-83-2R-IMPP is an inhibitor of PCSK9 translation. R-IMPP stimulates uptake of LDL-C in hepatoma cells by increasing LDL-R levels, without altering levels of secreted transferrin.
- $40
SizeQTY - CRT0066101 dihydrochlorideTQ01041883545-60-5CRT0066101 dihydrochloride is an effective and selective PKD inhibitor (IC50s: 1, 2.5 and 2 nM for PKD1, 2, and 3).
- $31
SizeQTY - SPHINX31T51941818389-84-2SPHINX31 is a potent inhibitor of serine/arginine-rich protein kinase 1 (SRPK1; IC50: 5.9 nM).
- $34
SizeQTY - 6-(Dimethylamino)purineT7444938-55-66-(Dimethylamino)purine (N,N-Dimethyladenine) is a serine threonine protein kinase and CDK inhibitor
- $29
SizeQTY - PCSK9-IN-10T72025368434-98-4PCSK9-IN-10, a potent and orally active inhibitor of Proprotein Convertase Subtilisin/Kexin Type 9 (PCSK9), exhibits a half-maximal inhibitory concentration (IC50) of 6.4 µM. By enhancing the expression of Low-Density Lipoprotein Receptor (LDLR) protein and reducing PCSK9 expression, PCSK9-IN-10 effectively decreases atherosclerosis progression. This compound holds promise for hyperlipidemia research applications.
- $41
SizeQTY - kb NB 142-70T20621233533-04-4kb NB 142-70 is a selective protein kinase D (PKD) inhibitor (IC50 values are 28.3, 58.7 and 53.2 nM for PKD1, 2 and 3 respectively).
- $40
SizeQTY - UpamostatT13257590368-25-5Upamostat is an inhibitor of a serine protease and is a urokinase plasminogen activator (uPA) inhibitor.
- $97
SizeQTY - PinostrobinTN2082480-37-5Pinostrobin, a potent flavonoid inducer, exerts a neuroprotective effect against Aα²(25-35)-induced neurotoxicity in PC12 cells, at least in part, via inhibiting oxidative damage and calcium overload, as well as suppressing the mitochondrial pathway of ce
- $81
SizeQTY - WNK-IN-11T54562123489-30-3WNK-IN-11 (Allosteric WNK Kinase Inhibitor) is an allosteric With-No-Lysine (WNK) kinase inhibitor,WNK1(IC50 : 4 nM)
- $84
SizeQTY - BioE-1115T105471268863-35-9BioE-1115 is a selective and potent inhibitor of serine-threonine protein kinase (PASK, IC50 = 4 nM). BioE-1115 is a potent inhibitor of CK2α (IC50 = 10 μM).
- $30
SizeQTY - WNK463T70172012607-27-9WNK463 is a pan-WNK-kinase inhibitor. It effectively inhibits the in vitro kinase activity of all four WNK family members (WNK1/2/3/4).
- $72
SizeQTY - Cetraxate hydrochlorideT1976327724-96-5Cetraxate hydrochloride (DV10062) is an oral gastrointestinal medication. It has a cytoprotective effect.
- $64
SizeQTY - FOY 251T867671079-09-9FOY 251 is a proteinase inhibitor, and is an anti-proteolytic active metabolite camostate.
- $49
SizeQTY - CID755673T2458521937-07-5CID755673 is an effective and specific cell-active inhibitor for PKD (IC50: 182 nM); exhibits selective PKD1 inhibition when compared with PLK1, AKT, CAMKIIα, CAK, and PKC isoforms.
- $35
SizeQTY - SGC-GAK-1T51692226517-76-4SGC-GAK-1 is a selective cyclin G-associated kinase (GAK) inhibitor (Ki: 3.1 nM).
- $31
SizeQTY - SRPIN340T1954218156-96-8SRPIN340 (SRPK inhibitor), a serine/arginine-rich protein kinase (SRPK)-specific inhibitor, is potent for SRPK1 (IC50 = 0.89 uM).
- $39
SizeQTY - kb-NB77-78T18081350622-33-1kb-NB77-78 is an analog of CID797718, which is a by-product of the synthesis of the parental compound, CID755673(PKD1 inhibitor).
- $47
SizeQTY - SBC-115076T2626489415-96-5SBC-115076 is a potent extracellular proprotein convertase subtilisin kexin type 9 (PCSK9) antagonist.
- $34
SizeQTY - ChymotrypsinT735949004-07-3Chymotrypsin (Chymotrypsin A) is a serine protease produced by the pancreas that cleaves protein chains on the carboxyl side of aromatic amino acids.
- $29
SizeQTY - SBC-110736T45241629166-02-4SBC-110736 is a proprotein convertase subtilisin kexin type 9 (PCSK9) inhibitor
- $48
SizeQTY - SM1-71T366802088179-99-9SM1-71 is a potent multi-targeted acrylamide-modified TAK1 inhibitor that inhibits MKNK2, MAP2K1/2/3/4/6/7, GAK, AAK1, BMP2K, MAP3K7, MAPKAPK5, GSK3A/B, MAPK1/3, SRC, YES1, FGFR1, ZAK (MLTK), MAP3K1, LIMK1 and RSK2.SM1-71 can be used as a kinase probe with anticancer activity and inhibits the proliferation of various cancer cell lines.
- $44
SizeQTY - Benzamidine hydrochlorideT83621670-14-0Benzamidine hydrochloride (Benzamidine HCl) is a reversible inhibitor of serine proteases, including trypsin, plasmin, and thrombin (Ki of 35, 350, and 220 μM, respectively).
- $40
SizeQTY
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