T11055 |
DL-TBOA
|
205309-81-5
|
98%
|
|
DL-TBOA inhibited [14C] glutamate uptake in COS-1 cells expressing human EAAT1 and EAAT2, with Ki values of 42 μM and 5.7 μM, respectively. DL-TBOA blocks EAAT4 ...
|
TN1033 |
Sennidin A
|
641-12-3
|
98%
|
|
Sennidin A, has two hydroxyanthraquinone-like moieties, exerts inhibition on NS3 helicase with IC50 values of 0.8 μM.
|
TN4288 |
Isoferulic acid
|
25522-33-2
|
98%
|
|
Isoferulic acid is an effective natural antioxidant in both lipid and aqueous media, it may be a new promising anti-glycation agent for the prevention of diabeti...
|
TN3885 |
Dodoviscin J
|
1372527-42-8
|
98%
|
|
Dodoviscin J can promote adipocyte differentiation as characterized by increased triglyceride levels in 3T3L1 cells.
|
TN1681 |
Gentianine
|
439-89-4
|
98%
|
|
Gentianine is an effective Swertiamarin derivative, which has anti-diabetic, antipsychotic, anti-inflammatory, hypotensive, diuretic and other effects, and has t...
|
TN3882 |
Dodoviscin A
|
1372527-25-7
|
98%
|
|
Dodoviscin A may be a new promising pigmentation-altering agent for cosmetic and therapeutic applications, it can inhibit melanin biosynthesis induced by 3-isobu...
|
TMA0127 |
Ficusin A
|
173429-83-9
|
98%
|
|
Ficusin has antioxidant, antilipidemic and antidiabetic effects, it can lower the levels of fasting blood glucose, plasma insulin, body weight gain in HFD-STZ in...
|
T13330L |
WAY-213613
|
868359-05-1
|
98%
|
|
WAY-213613 is a potent and selective nonsubstrate reuptake inhibitor of GLT-1/EAAT2 (IC50: 85 nM EAAT2). It displays 59- and 44-fold selectivity over EAAT1 and E...
|
TN3884 |
Dodoviscin I
|
1372527-40-6
|
98%
|
|
Dodoviscin I can promote adipocyte differentiation as characterized by increased triglyceride levels in 3T3L1 cells.
|
TN2535 |
1-Hydroxy-2-oxopomolic acid
|
217466-37-0
|
98%
|
|
1β-Hydroxy-2-oxopomolic acid inhibits adipocyte differentiation through downregulation of various adipocytokines by blocking PPARγ and C/EBPα expression.
|
TN1034 |
Sennidin B
|
517-44-2
|
98%
|
|
Sennidin B stimulates glucose incorporation in rat adipocytes.
|
TN3883 |
Dodoviscin H
|
1372527-39-3
|
98%
|
|
Dodoviscin H can promote adipocyte differentiation as characterized by increased triglyceride levels in 3T3L1 cells.
|
T40083 |
GLUT inhibitor-1
|
2421141-40-2
|
98%
|
|
GLUT inhibitor-1 is an orally active GLUT inhibitor with IC50 s of 242 nM and 179 nM for GLUT1 and GLUT3. GLUT inhibitor-1 can be used in studies about cancers a...
|
T4182 |
Lavendustin B
|
125697-91-8
|
95.72%
|
|
Lavendustin B is a Tyrosine Kinase Inhibitor and an inhibitor of HIV-1 integrase (IN) interaction with its cognate cellular cofactor, lens epithelium-derived gro...
|
T4138 |
UCPH-101
|
1118460-77-7
|
98%
|
|
UCPH-101 is an inhibitor of excitatory amino acid transporter subtype 1 (EAAT1) with an IC50 of 0.66 μM.
|
T4S1545 |
Licarin B
|
51020-87-2
|
98%
|
|
1.(-)-Licarin B has anti-mycobacterial activity.
|
T2755 |
Rhoifolin
|
17306-46-6
|
98.11%
|
|
Rhoifolin is extracted from Turpinia arguya Seem dried leaves.
|
T15728 |
LDN-212320
|
894002-50-7
|
98.13%
|
|
LDN-212320 is a glutamate transporter EAAT2 activator. It also enhances EAAT2 levels by > 6 fold at concentrations < 5 μM after 24 h.
|
T22317 |
DRB18
|
T22317
|
98.74%
|
|
DRB18 is a potent pan-class GLUT inhibitor. DRB18 alters energy-related metabolism in A549 cells by changing the abundance of metabolites in glucose-related path...
|
TN1132 |
Procyanidin A2
|
41743-41-3
|
98.78%
|
|
Procyanidin A2 is a potential precursor of 5-(3',4'-dihydroxyphenyl)-γ-valerolactone, exhibits antioxidant, anti-inflammary, anti-hyperglycemia, and anti-type 2 ...
|