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Troriluzole
🥰Excellent
Catalog No. T17174Cas No. 1926203-09-9
Alias FC 4157, BHV-4157a, BHV-4157, BHV4157, BHV 4157
Troriluzole is an orally active glutamate modulator with anticancer activity.Troriluzole enhances the expression of excitatory amino acid transporters located in glial cells and is used in the study of spinocerebellar ataxia, Alzheimer's disease, and generalized anxiety disorder (GAD).
Troriluzole
🥰Excellent
Purity: 97.14%
Catalog No. T17174Alias FC 4157, BHV-4157a, BHV-4157, BHV4157, BHV 4157Cas No. 1926203-09-9
Troriluzole is an orally active glutamate modulator with anticancer activity.Troriluzole enhances the expression of excitatory amino acid transporters located in glial cells and is used in the study of spinocerebellar ataxia, Alzheimer's disease, and generalized anxiety disorder (GAD).
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $100 | In Stock | |
| 5 mg | $247 | In Stock | |
| 10 mg | $396 | In Stock | |
| 25 mg | $728 | In Stock | |
| 50 mg | $1,160 | In Stock | |
| 100 mg | $1,730 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $272 | In Stock |
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CitedSelect Batch
Purity:97.14%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Troriluzole is an orally active glutamate modulator with anticancer activity.Troriluzole enhances the expression of excitatory amino acid transporters located in glial cells and is used in the study of spinocerebellar ataxia, Alzheimer's disease, and generalized anxiety disorder (GAD). |
| In vitro | Troriluzole is an EAAT2 modulator, NMDA receptor antagonist, and Nav1.5 blocker, commonly used in research on neurological disorders such as obsessive-compulsive disorder[1]. |
| Alias | FC 4157, BHV-4157a, BHV-4157, BHV4157, BHV 4157 |
| Molecular Weight | 419.38 |
| Formula | C15H16F3N5O4S |
| Cas No. | 1926203-09-9 |
| Smiles | CN(CC(=O)Nc1nc2ccc(OC(F)(F)F)cc2s1)C(=O)CNC(=O)CN |
| Relative Density. | 1.518 g/cm3 (Predicted) |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 30 mg/mL (71.53 mM), Sonication is recommended. | ||||||||||||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||||||||||||
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
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