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Biochemicals
- Autophagy
- Cell Cycle/Checkpoint
- Cytoskeletal Signaling
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- IDO
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- E3 Ligase Ligand-Linker Conjugate
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- Tumor
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- Other Fields
- Alangiaceae
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- Cephalotaxaceae
- Costaceae
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- Dioscoreaceae
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- Hematologic Malignancies Target Proteins
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- Hydrolases,EC 3
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- Ligases or Synthetases,EC 6
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- Coronavirus (CoV) Proteins
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- HIV Proteins
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- Molecular Docking
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Cell Cycle/CheckpointHaspin Kinase
Serine/threonine-protein kinase haspin is an enzyme that in humans is encoded by the GSG2 gene.
AZ1495
T143672196204-23-4
AZ1495 is an oral active inhibitor of Interleukin-1 receptor associated kinase 4 (IRAK4), with IC50 values of 5 nM and 23 nM for IRAK4 and IRAK1, respectively. Which Shows activity in treatment of mutant MYD88L265P diffuse large B-cell lymphoma (DLBCL).
- $148
Size
QTY
LDN-192960
TQ0111184582-62-5
LDN-192960 is a potent inhibitor of Haspin and DYRK2 (IC50s: 10 nM and 48 nM).
- $133
Size
QTY
Haspin-IN-3
T605122416569-95-2
Haspin-IN-3 is a potent haspin inhibitor with an IC50 of 14 nM.Haspin-IN-3 has anticancer activity.
- $60
Size
QTY
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