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Imepitoin

Catalog No. T1860Cas No. 188116-07-6
Alias ELB-138, AWD 131-138

Imepitoin (AWD 131-138) is a novel low-affinity partial benzodiazepine receptor agonist, exhibiting potent anticonvulsant and anxiolytic properties in rodent models.

Imepitoin

Imepitoin

Purity: 98.45%
Catalog No. T1860Alias ELB-138, AWD 131-138Cas No. 188116-07-6
Imepitoin (AWD 131-138) is a novel low-affinity partial benzodiazepine receptor agonist, exhibiting potent anticonvulsant and anxiolytic properties in rodent models.
Pack SizePriceAvailabilityQuantity
2 mg$31In Stock
5 mg$48In Stock
10 mg$85In Stock
25 mg$172In Stock
50 mg$289In Stock
100 mg$419In Stock
1 mL x 10 mM (in DMSO)$54In Stock
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Purity:98.45%
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Product Introduction

Bioactivity
Description
Imepitoin (AWD 131-138) is a novel low-affinity partial benzodiazepine receptor agonist, exhibiting potent anticonvulsant and anxiolytic properties in rodent models.
Kinase Assay
Cell-based determinations of mTOR inhibition: A high-throughput screening cell-based assay is developed using MDA-MB-468 cells to detect mTORC1 and mTORC2 activity. Cells are exposed for 2 hours to increasing concentrations of AZD8055. At the end of the incubation period, cells are fixed, washed, and probed with antibodies against S473 pAkt or against S235/236 phosphorylated S6 (pS6). Levels of phosphorylation are assessed using an Acumen laser scanning cytometer.
AliasELB-138, AWD 131-138
Chemical Properties
Molecular Weight279.72
FormulaC13H14ClN3O2
Cas No.188116-07-6
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
DMSO: 13 mg/mL (46.48 mM), Sonication is recommended.
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM3.5750 mL17.8750 mL35.7500 mL178.7502 mL
5 mM0.7150 mL3.5750 mL7.1500 mL35.7500 mL
10 mM0.3575 mL1.7875 mL3.5750 mL17.8750 mL
20 mM0.1788 mL0.8938 mL1.7875 mL8.9375 mL

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Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
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