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AR-M 1896 Acetate

AR-M 1896 Acetate
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Purity:95.32%
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AR-M 1896 Acetate

Catalog No. T21646L
AR-M 1896 Acetate is the selective agonist of GalR2.
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Pack SizePriceAvailabilityQuantity
1 mg$941In Stock
5 mg$1,880In Stock
10 mg$2,560In Stock
25 mg$3,780In Stock
50 mg$5,130In Stock
100 mg$6,920In Stock
1 mL x 10 mM (in DMSO)$3,910In Stock
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Product Introduction

Bioactivity
Description
AR-M 1896 Acetate is the selective agonist of GalR2.
In vitro
Removal of the glycine residue in position 1 resulted in AR-M1896 with almost unchanged GalR2 affinity and functional activity, and 500-fold selectivity for GalR2-Rs over GalR1-Rs[1].?
In vivo
In normal rats mechanical and cold allodynia of the hindpaw are induced by intrathecal infusion of low-dose galanin. The same effect is seen with equimolar doses of AR-M1896 or AR-M961 (an agonist both at GalR1 and GalR2 receptors). In allodynic Bennett model rats, the mechanical threshold dose-dependently increased after intrathecal injection of a high AR-M961dose, whereas no effect was observed in the control or AR-M1896 group. No effect of either compounds was observed in nonallodynic Bennett model rats[1].
AliasAR-M 1896 Acetate (367518-31-8 Free base)
Chemical Properties
Molecular Weight1196.35
FormulaC56H85N13O16
Cas No.
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year
Solubility Information
DMSO: 55 mg/ml (45.97 mM)
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM0.8359 mL4.1794 mL8.3588 mL41.7938 mL
5 mM0.1672 mL0.8359 mL1.6718 mL8.3588 mL
10 mM0.0836 mL0.4179 mL0.8359 mL4.1794 mL
20 mM0.0418 mL0.2090 mL0.4179 mL2.0897 mL

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