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ML-354
🥰Excellent
Catalog No. T21901Cas No. 89159-60-4
Alias VU0099704, VU 0099704, ML354
ML-354 (VU0099704) is a selective and potent PAR4 antagonist for the study of cardiovascular disease.
ML-354
🥰Excellent
Catalog No. T21901Alias VU0099704, VU 0099704, ML354Cas No. 89159-60-4
ML-354 (VU0099704) is a selective and potent PAR4 antagonist for the study of cardiovascular disease.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $50 | In Stock | |
| 5 mg | $113 | In Stock | |
| 10 mg | $197 | In Stock | |
| 25 mg | $462 | In Stock | |
| 50 mg | $669 | In Stock | |
| 100 mg | $943 | In Stock | |
| 200 mg | $1,270 | In Stock |
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Product Introduction
Bioactivity
Chemical Properties
| Description | ML-354 (VU0099704) is a selective and potent PAR4 antagonist for the study of cardiovascular disease. |
| Targets&IC50 | PAR4 receptor:140 nM |
| In vitro | ML-354 is a specific PAR4 receptor antagonist with an IC50 value of 140 nM. [1] |
| Alias | VU0099704, VU 0099704, ML354 |
| Molecular Weight | 282.29 |
| Formula | C16H14N2O3 |
| Cas No. | 89159-60-4 |
| Smiles | CN1C(CO)=C(C2=CC=CC=C2)C3=C1C=CC([N+]([O-])=O)=C3 |
| Relative Density. | 1.29g/cm3 |
Storage & Solubility Information
| Storage | store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 20 mg/mL (70.85 mM), Sonication is recommended. | ||||||||||||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||||||||||||
DMSO
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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