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AY 77
🥰Excellent
Catalog No. T41190Cas No. 1835734-92-3
Alias Unk-Cha-Chg-NH2
AY 77 (Unk-Cha-Chg-NH2) is a potent and selective PAR2 agonist. AY 77 showed selectivity for Ca2+ and ERK1/2 signaling (ec50 value of Ca2+ release was 40 nM and ec50 value of ERK1/2 phosphorylation was 2 μM). AY 77 can promote migration of human breast cancer cells in vitro.
AY 77
🥰Excellent
Purity: 99.7%
Catalog No. T41190Alias Unk-Cha-Chg-NH2Cas No. 1835734-92-3
AY 77 (Unk-Cha-Chg-NH2) is a potent and selective PAR2 agonist. AY 77 showed selectivity for Ca2+ and ERK1/2 signaling (ec50 value of Ca2+ release was 40 nM and ec50 value of ERK1/2 phosphorylation was 2 μM). AY 77 can promote migration of human breast cancer cells in vitro.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $412 | In Stock | |
| 5 mg | $888 | In Stock | |
| 10 mg | $1,190 | In Stock | |
| 25 mg | $1,770 | In Stock | |
| 50 mg | $2,390 | In Stock | |
| 100 mg | $3,230 | In Stock |
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Purity:99.7%
ee:100%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | AY 77 (Unk-Cha-Chg-NH2) is a potent and selective PAR2 agonist. AY 77 showed selectivity for Ca2+ and ERK1/2 signaling (ec50 value of Ca2+ release was 40 nM and ec50 value of ERK1/2 phosphorylation was 2 μM). AY 77 can promote migration of human breast cancer cells in vitro. |
| Alias | Unk-Cha-Chg-NH2 |
| Molecular Weight | 404.5 |
| Formula | C21H32N4O4 |
| Cas No. | 1835734-92-3 |
| Smiles | [C@H](CC1CCCCC1)(C(N[C@H](C(N)=O)[C@@H]2CCCCC2)=O)NC(=O)C3=CC=NO3 |
| Relative Density. | 1.183 g/cm3 (Predicted) |
Storage & Solubility Information
| Storage | keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||
| Solubility Information | Ethanol: 0.9 mg/mL (2.2 mM) | ||||||||||
Solution Preparation Table | |||||||||||
Ethanol
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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