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AY 77
Contact us for more batch information
AY 77
Catalog No. T41190Cas No. 1835734-92-3
AY 77 (Unk-Cha-Chg-NH2) is a potent and selective PAR2 agonist. AY 77 showed selectivity for Ca2+ and ERK1/2 signaling (ec50 value of Ca2+ release was 40 nM and ec50 value of ERK1/2 phosphorylation was 2 μM). AY 77 can promote migration of human breast cancer cells in vitro.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $686 | In Stock | |
| 5 mg | $1,480 | In Stock | |
| 10 mg | $1,990 | In Stock | |
| 25 mg | $2,960 | In Stock | |
| 50 mg | $3,990 | In Stock | |
| 100 mg | $5,390 | In Stock |
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Product Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | AY 77 (Unk-Cha-Chg-NH2) is a potent and selective PAR2 agonist. AY 77 showed selectivity for Ca2+ and ERK1/2 signaling (ec50 value of Ca2+ release was 40 nM and ec50 value of ERK1/2 phosphorylation was 2 μM). AY 77 can promote migration of human breast cancer cells in vitro. |
| Alias | Unk-Cha-Chg-NH2 |
| Molecular Weight | 404.5 |
| Formula | C21H32N4O4 |
| Cas No. | 1835734-92-3 |
| Storage | keep away from moisture Powder: -20°C for 3 years | In solvent: -80°C for 1 year | ||||||||||||||||||||||||||||||
| Solubility Information | Ethanol: 0.9 mg/mL (2.2 mM) | ||||||||||||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||||||||||||
Ethanol
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