Shopping Cart
- Remove All
Your shopping cart is currently empty
MRGPRX1 agonist 1
Catalog No. T12104Cas No. 2377379-39-8
MRGPRX1 agonist 1 is a highly potent agonist of MRGPRX1 (Mas-related G-protein-coupled receptor X1) with an EC50 of 50 nM.
MRGPRX1 agonist 1
Catalog No. T12104Cas No. 2377379-39-8
MRGPRX1 agonist 1 is a highly potent agonist of MRGPRX1 (Mas-related G-protein-coupled receptor X1) with an EC50 of 50 nM.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $90 | In Stock | |
| 5 mg | $222 | In Stock | |
| 10 mg | $355 | In Stock | |
| 25 mg | $645 | In Stock | |
| 50 mg | $883 | In Stock | |
| 100 mg | $1,260 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $245 | In Stock |
Bulk & Custom
Add to Cart
Questions
View MoreInhibitors Related to "MRGPRX1 agonist 1"
BAM (8-22) acetate
BAM (8-22) acetate(412961-36-5 free base)
TP1914L1
BAM (8-22) acetate is a proteolytically cleaved product of proenkephalin A. BAM (8-22) acetate activates Mas-related G-protein-coupled receptors (Mrgprs), MrgprC11 and hMrgprX1, and induces scratching in mice in an Mrgpr-dependent manner.
- $319
Size
QTY
(R)-ZINC-3573
ZINC 3573
T292212089389-15-9
(R)-ZINC-3573 is a potent and highly selective MRGPRX2 probe that activates endogenous MRGPRX2 in a human mast cell line, inducing degranulation and calcium release.
- $39
Size
QTY
ML382
T85381646499-97-9
ML382 is a potent and selective MrgX1 positive allosteric modulator (EC50 : 190 nM).
- $41
Size
QTY
MrgprX2 antagonist-8
T638122768216-96-0
MrgprX2 antagonist-8 is an MrgprX2 antagonist that can be used to study inflammatory diseases.
- $106
Size
QTY
MRGPRX4 modulator-2
T611832492595-24-9
MRGPRX4 modulator-2 (compound 1-55) is a highly potent antagonist of MRGPRX4 with an IC50 value of less than 100 nM. Its notable applications include research on autoimmune diseases such as psoriasis, multiple sclerosis, Steven Johnson's Syndrome, and various chronic itch conditions [1].
- $52
Size
QTY
Select Batch
Purity:99.59%
Contact us for more batch information
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | MRGPRX1 agonist 1 is a highly potent agonist of MRGPRX1 (Mas-related G-protein-coupled receptor X1) with an EC50 of 50 nM. |
| Targets&IC50 | MRGPRX1:50 nM(EC50) |
| Molecular Weight | 435.5 |
| Formula | C23H21N3O4S |
| Cas No. | 2377379-39-8 |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 125 mg/mL (287.03 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
| ||||||||||||||||||||||||||||||||||||
Calculator
In Vivo Formulation Calculator (Clear solution)
Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . A total of 10 animals were administered, and the formula you used is 5% 
DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
Dose Conversion
You can also refer to dose conversion for different animals. More Dose Conversion
Tech Support
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc
Preview
Related Tags: buy MRGPRX1 agonist 1 | purchase MRGPRX1 agonist 1 | MRGPRX1 agonist 1 cost | order MRGPRX1 agonist 1 | MRGPRX1 agonist 1 chemical structure | MRGPRX1 agonist 1 formula | MRGPRX1 agonist 1 molecular weight
- TOP
Feedback
Hello! How can I help you today? 
Copyright © 2015-2024 TargetMol Chemicals Inc. All Rights Reserved.