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NS-102
🥰Excellent
Catalog No. T38779Cas No. 136623-01-3
Alias NS102, NS 102
NS-102 is a glutamate receptor and NMDA receptor antagonist that inhibits erythrocyanine (GluK2), which reduces glur6 receptor-mediated currents, and inhibits specific binding to the glur6 receptor.
NS-102
🥰Excellent
Purity: 98.95%
Catalog No. T38779Alias NS102, NS 102Cas No. 136623-01-3
NS-102 is a glutamate receptor and NMDA receptor antagonist that inhibits erythrocyanine (GluK2), which reduces glur6 receptor-mediated currents, and inhibits specific binding to the glur6 receptor.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $158 | In Stock | |
| 5 mg | $396 | In Stock | |
| 10 mg | $662 | In Stock | |
| 25 mg | $1,090 | In Stock | |
| 50 mg | $1,470 | In Stock | |
| 100 mg | $1,980 | In Stock |
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Purity:98.95%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | NS-102 is a glutamate receptor and NMDA receptor antagonist that inhibits erythrocyanine (GluK2), which reduces glur6 receptor-mediated currents, and inhibits specific binding to the glur6 receptor. |
| In vitro | NS-102, an AMPA receptor antagonist, when used in combination with GYKI 52466 (30 μM) at a concentration of 10 μM, prevents complete loss of compound action potentials (CAP) during oxygen and glucose deprivation (OGD), and enhances the recovery of CAP amplitude [1]. |
| In vivo | NS-102 (20, 40, or 80 μmol/litre; in the hippocampal CA3 region) significantly reduces Sevoflurane-induced hyperactivities[1]. |
| Alias | NS102, NS 102 |
| Molecular Weight | 261.23 |
| Formula | C12H11N3O4 |
| Cas No. | 136623-01-3 |
| Smiles | O\N=C1/C(=O)Nc2c1cc(c1CCCCc21)[N+]([O-])=O |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||
| Solubility Information | DMSO: 2 mg/mL (7.6 mM), Sonication is recommended. | |||||||||||||||
Solution Preparation Table | ||||||||||||||||
DMSO
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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