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PROTAC BRD4 ligand-1

PROTAC BRD4 ligand-1
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Purity:99.48%
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PROTAC BRD4 ligand-1

Catalog No. T12551Cas No. 2313230-51-0
PROTAC BRD4 ligand-1 is a ligand for PROTAC GNE-987 targeting the BRD4 protein and is an inhibitor of BET.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.
Pack SizePriceAvailabilityQuantity
1 mg$125In Stock
5 mg$313In Stock
10 mg$522In Stock
25 mg$987In Stock
50 mg$1,660In Stock
100 mg$2,390In Stock
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Product Introduction

Bioactivity
Description
PROTAC BRD4 ligand-1 is a ligand for PROTAC GNE-987 targeting the BRD4 protein and is an inhibitor of BET.
Chemical Properties
Molecular Weight500.47
FormulaC23H18F2N4O5S
Cas No.2313230-51-0
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year
Solubility Information
DMSO: 4.5 mg/mL (9.0 mM)
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM1.9981 mL9.9906 mL19.9812 mL99.9061 mL
5 mM0.3996 mL1.9981 mL3.9962 mL19.9812 mL

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TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
1 Enter information below:
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

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