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PROTAC EZH2 Degrader-1
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Catalog No. T74602Cas No. 2641601-67-2
PROTAC EZH2 Degrader-1 (Compound 150d) is a potent inhibitor that effectively suppresses EZH2 methyltransferase activity, with an IC50 of 2.7 nM. EZH2 plays a critical role in various tumorigenesis and development processes [1].
PROTAC EZH2 Degrader-1
😃Good
Catalog No. T74602Cas No. 2641601-67-2
PROTAC EZH2 Degrader-1 (Compound 150d) is a potent inhibitor that effectively suppresses EZH2 methyltransferase activity, with an IC50 of 2.7 nM. EZH2 plays a critical role in various tumorigenesis and development processes [1].
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $215 | 7-10 days | |
| 5 mg | $645 | 7-10 days | |
| 10 mg | $975 | 7-10 days |
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Product Introduction
Bioactivity
Chemical Properties
| Description | PROTAC EZH2 Degrader-1 (Compound 150d) is a potent inhibitor that effectively suppresses EZH2 methyltransferase activity, with an IC50 of 2.7 nM. EZH2 plays a critical role in various tumorigenesis and development processes [1]. |
| Molecular Weight | 942.15 |
| Formula | C54H67N7O8 |
| Cas No. | 2641601-67-2 |
Storage & Solubility Information
| Storage | Shipping with blue ice. |
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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