Shopping Cart
  • Remove All
  • TargetMol
    Your shopping cart is currently empty

PSB-12379 ditriethylamine salt

🥰Excellent
Catalog No. T12569L

PSB-12379 ditriethylamine salt, a nucleotide analogue, is a potent Ecto-5'-Nucleotidase (CD73) inhibitor with Kis of 9.03 nM (rat) and 2.21 nM (human).

PSB-12379 ditriethylamine salt

PSB-12379 ditriethylamine salt

🥰Excellent
Purity: 99.75%
Catalog No. T12569L
PSB-12379 ditriethylamine salt, a nucleotide analogue, is a potent Ecto-5'-Nucleotidase (CD73) inhibitor with Kis of 9.03 nM (rat) and 2.21 nM (human).
Pack SizePriceAvailabilityQuantity
1 mg$70In Stock
5 mg$161In Stock
10 mg$237In Stock
25 mg$355In Stock
50 mg$500In Stock
100 mg$672In Stock
200 mg$890In Stock
1 mL x 10 mM (in DMSO)$231In Stock
Bulk & Custom
Add to Cart
Questions
View More

Related Compound Libraries of "PSB-12379 ditriethylamine salt"

Select Batch
Purity:99.75%
Contact us for more batch information
Resource Download
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

Product Introduction

Bioactivity
Description
PSB-12379 ditriethylamine salt, a nucleotide analogue, is a potent Ecto-5'-Nucleotidase (CD73) inhibitor with Kis of 9.03 nM (rat) and 2.21 nM (human).
In vitro
Metabolism: Only a small percentage (<23%) of PSB-12379 (10g) is metabolized under the applied conditions, while >77% of the compounds are recovered unchanged after a long incubation for 8 h. PSB-12379 (10g) is somewhat less stable, and 56% are metabolized within 8 h. Hydrolytic cleavage of the glycosidic bond, which is a typical phase I reaction of nucleosides and nucleotides, was observed as the main reaction[1].
Chemical Properties
Molecular Weight717.73
FormulaC30H53N7O9P2
SmilesO=P(CP(O)(O)=O)(O)OC[C@@H](O1)[C@@H](O)[C@@H](O)[C@@H]1N2C3=NC=NC(NCC4=CC=CC=C4)=C3N=C2.CCN(CC)CC.CCN(CC)CC
Relative Density.no data available
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
DMSO: 11 mg/mL (15.33 mM)
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM1.3933 mL6.9664 mL13.9328 mL69.6641 mL
5 mM0.2787 mL1.3933 mL2.7866 mL13.9328 mL
10 mM0.1393 mL0.6966 mL1.3933 mL6.9664 mL

Calculator

  • Molarity Calculator
  • Dilution Calculator
  • Reconstitution Calculator
  • Molecular Weight Calculator

In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
1 Enter information below:
mg/kg
g
μL
2 Enter the in vivo formulation:
% DMSO
%
%Tween 80
%ddH2O

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

Related Tags: buy PSB-12379 ditriethylamine salt | purchase PSB-12379 ditriethylamine salt | PSB-12379 ditriethylamine salt cost | order PSB-12379 ditriethylamine salt | PSB-12379 ditriethylamine salt chemical structure | PSB-12379 ditriethylamine salt in vitro | PSB-12379 ditriethylamine salt formula | PSB-12379 ditriethylamine salt molecular weight