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SLF-amido-C2-COOH
🥰Excellent
Catalog No. T13914Cas No. 1092369-24-8
Alias PROTAC FKBP12-binding moiety 1
SLF-amido-C2-COOH (ZZY01-083) is an FKBP ligand with potential antimicrobial activity for the synthesis of PROTAC.
SLF-amido-C2-COOH
🥰Excellent
Catalog No. T13914Alias PROTAC FKBP12-binding moiety 1Cas No. 1092369-24-8
SLF-amido-C2-COOH (ZZY01-083) is an FKBP ligand with potential antimicrobial activity for the synthesis of PROTAC.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $65 | In Stock | |
| 5 mg | $157 | In Stock | |
| 10 mg | $267 | In Stock | |
| 25 mg | $593 | In Stock |
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Product Introduction
Bioactivity
Chemical Properties
| Description | SLF-amido-C2-COOH (ZZY01-083) is an FKBP ligand with potential antimicrobial activity for the synthesis of PROTAC. |
| In vitro | SLF-amido-C2-COOH is a synthetic ligand (SLF) that binds FKBP.SLF consists of a portion of the structure of FK506 and has a relatively weak binding capacity to FKBP12. [1] |
| Alias | PROTAC FKBP12-binding moiety 1 |
| Molecular Weight | 624.72 |
| Formula | C34H44N2O9 |
| Cas No. | 1092369-24-8 |
| Smiles | [C@@H](OC(=O)[C@H]1N(C(C(C(CC)(C)C)=O)=O)CCCC1)(CCC2=CC(OC)=C(OC)C=C2)C3=CC(NC(CCC(O)=O)=O)=CC=C3 |
| Relative Density. | 1.225 g/cm3 (Predicted) |
Storage & Solubility Information
| Storage | keep away from direct sunlight,store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 80 mg/mL (128.06 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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